SCHEMBL28826953

SCHEMBL28826953

CC(C)(C)C1C(Oc2cccc(N)c2)CCCN1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
CPT1A P50416 1/20 0.37
OPRK1 P41145 3/20 0.36
KCNH2 Q12809 1/20 0.36
CHRM3 P20309 3/20 0.36
ALDH1A1 P00352 2/20 0.36
RIPK1 Q13546 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LTA4H P09960 1/20 0.36
MAOB P27338 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPK1 P28482 1/20 0.35
LMNA P02545 1/20 0.34
DPP4 P27487 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28059288 0.93 OPRK1 (0.38) POLBCHRNB2CHRNA4CPT1AOPRK1
SCHEMBL28059300 0.86 CHRM3 (0.38) POLBCHRNB2CHRNA4OPRK1KCNH2
SCHEMBL20658831 0.77 TSHR (0.38) POLBOPRK1KCNH2CHRM3ALDH1A1
SCHEMBL28053867 0.76 OPRK1 (0.41) POLBOPRK1KCNH2CHRM3
SCHEMBL4279118 0.76 CHRM3 (0.36) OPRK1KCNH2CHRM3
SCHEMBL4279130 0.76 CHRM3 (0.36) OPRK1KCNH2CHRM3
SCHEMBL28059315 0.76 SLC6A2 (0.44) CHRNB2CHRNA4CPT1AALDH1A1LTA4H
SCHEMBL23582990 0.73 RIPK1 (0.38) ALDH1A1RIPK1LMNADPP4DPP8
SCHEMBL23582028 0.73 TSHR (0.48)
SCHEMBL23526972 0.70 EPHX2 (0.42) ALDH1A1LMNANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384695-A Pyrimidine derivative, preparation method therefor and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed