SCHEMBL28061819

SCHEMBL28061819

O=c1c2ccccc2ccn1Cc1cccc(Br)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
KMT2A Q03164 2/20 0.46
CYP19A1 P11511 1/20 0.46
HPGD P15428 1/20 0.46
ACHE P22303 1/20 0.45
CYP11B1 P15538 1/20 0.44
ADRA2C P18825 1/20 0.44
CYP11B2 P19099 1/20 0.44
DRD4 P21917 1/20 0.44
NLRP3 Q96P20 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061870 0.84 CNR2 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL29809414 0.83 ACHE (0.59) KMT2AACHEDHPSKDM4EMEN1
SCHEMBL1757848 0.83 ACHE (0.59) KMT2AACHEDHPSKDM4EMEN1
SCHEMBL28061820 0.83 MAPT (0.58) KMT2AACHECYP11B1CYP11B2DRD4
SCHEMBL13392342 0.81 PSMB1 (0.48) KMT2AACHEDHPSMEN1ALDH1A1
SCHEMBL31241086 0.81 PSMB1 (0.48) KMT2AACHEDHPSMEN1ALDH1A1
SCHEMBL2120980 0.81 MAPK14 (0.48) KMT2AACHEIDO1DHPSMEN1
SCHEMBL30218821 0.79 HTR6 (0.55) HDAC1HDAC2HDAC10HDAC8HDAC6
SCHEMBL6086304 0.79 HTR6 (0.55) HDAC1HDAC2HDAC10HDAC8HDAC6
SCHEMBL6171027 0.79 EGLN1 (0.53) KMT2AKDM4EALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503724-B A kind of preparation method of the polysubstituted compound of isobioquin group of 2 benzyl 1 湘潭大学 2018-01-30 CN disclosed
CN-105503724-A Preparation method of polysubstituted 2-benzyl-1-isoquinolone compound UNIV XIANGTAN 2016-04-20 CN disclosed