SCHEMBL28061870

SCHEMBL28061870

O=c1c2ccccc2ccn1Cc1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.49
ACHE P22303 1/20 0.48
KMT2A Q03164 5/20 0.47
MEN1 O00255 3/20 0.47
HTT P42858 1/20 0.47
PLAU P00749 1/20 0.44
GAA P10253 2/20 0.44
MGAM O43451 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC11 Q96DB2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29809414 0.87 ACHE (0.59) ACHEKMT2AMEN1HTTALDH1A1
SCHEMBL1757848 0.87 ACHE (0.59) ACHEKMT2AMEN1HTTALDH1A1
SCHEMBL5183061 0.84 MAPT (0.55) CNR2ACHEKMT2AMEN1HTT
SCHEMBL28061855 0.84 MAPT (0.62) ACHEKMT2AMEN1HTTGAA
SCHEMBL31667042 0.84 NLRP3 (0.49) ACHEKMT2AMEN1HTTPLAU
SCHEMBL28061819 0.84 HDAC3 (0.47) ACHEKMT2AMEN1HDAC1HDAC2
SCHEMBL2120980 0.82 MAPK14 (0.48) ACHEKMT2AMEN1GAAALDH1A1
SCHEMBL31241086 0.82 PSMB1 (0.48) ACHEKMT2AMEN1GAAALDH1A1
SCHEMBL13392342 0.82 PSMB1 (0.48) ACHEKMT2AMEN1GAAALDH1A1
SCHEMBL28525032 0.81 KDM4E (0.47) ACHEKMT2AHTTHDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503724-B A kind of preparation method of the polysubstituted compound of isobioquin group of 2 benzyl 1 湘潭大学 2018-01-30 CN disclosed
CN-105503724-A Preparation method of polysubstituted 2-benzyl-1-isoquinolone compound UNIV XIANGTAN 2016-04-20 CN disclosed