SCHEMBL28065527

SCHEMBL28065527

Nc1nc2ccccc2nc1-c1c[c]ccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 5/20 0.47
GAA P10253 4/20 0.47
HSD17B10 Q99714 3/20 0.47
MAPT P10636 3/20 0.47
HPGD P15428 2/20 0.47
KMT2A Q03164 3/20 0.39
ATM Q13315 1/20 0.39
TLR9 Q9NR96 1/20 0.39
PKM P14618 2/20 0.38
LMNA P02545 4/20 0.37
L3MBTL1 Q9Y468 4/20 0.37
TDP1 Q9NUW8 3/20 0.37
MEN1 O00255 2/20 0.37
CSNK1A1 P48729 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
ADORA2A P29274 3/20 0.36
NUDT1 P36639 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21382895 0.84 KDM4E (0.53) KDM4EALDH1A1GAAHPGDKMT2A
SCHEMBL28828233 0.79 KDM4E (0.65) KDM4EALDH1A1GAAMAPTKMT2A
SCHEMBL384076 0.79 KDM4E (0.61) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL28600927 0.76 NUDT1 (0.43) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL29215313 0.72 KDM4E (0.56) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL225976 0.70 SMN1; SMN2 (0.37) KDM4EALDH1A1MAPTHPGDLMNA
SCHEMBL31448436 0.69 TDP1 (0.69) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL1450354 0.69 NPC1 (0.53) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL23625965 0.68 SRC (0.51) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL28586210 0.68 ESR1 (0.51) KDM4EALDH1A1GAAHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683182-A Biaryl acetamide compounds and methods of use thereof 埃姆比特生物科学公司 2016-06-15 CN disclosed