SCHEMBL28066927

SCHEMBL28066927

Nc1ncc(-c2ccc(N3CCNCC3)cc2)c(NCC2CCCO2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 12/20 0.60
ALDH1A1 P00352 2/20 0.48
CYP1A2 P05177 1/20 0.48
MAPT P10636 1/20 0.48
CYP2C19 P33261 1/20 0.48
HTT P42858 1/20 0.48
CHEK1 O14757 1/20 0.47
JAK2 O60674 1/20 0.47
ABL1 P00519 1/20 0.47
LCK P06239 1/20 0.47
ROS1 P08922 1/20 0.47
FGFR1 P11362 1/20 0.47
SRC P12931 1/20 0.47
TYK2 P29597 1/20 0.47
ALK Q9UM73 1/20 0.47
SYK P43405 5/20 0.45
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28066917 0.91 TNK2 (0.58) TNK2ALDH1A1MAPTCHEK1JAK2
SCHEMBL28066957 0.89 TNK2 (0.60) TNK2ALDH1A1CYP1A2CHEK1JAK2
SCHEMBL28829103 0.79 TNK2 (0.53) TNK2ALDH1A1CYP1A2MAPTCYP2C19
SCHEMBL16453378 0.75 TNK2 (1.00) TNK2CHEK1JAK2ABL1LCK
SCHEMBL16447803 0.74 TNK2 (1.00) TNK2CHEK1JAK2ABL1LCK
Hydrochloric Acid SCHEMBL28067024 0.74 L3MBTL1 (0.45) TNK2ALDH1A1CYP1A2MAPTCYP2C19
SCHEMBL30515653 0.72 DHFR (0.56)
SCHEMBL17907560 0.72 DHFR (0.56)
SCHEMBL1588124 0.70 HRH4 (0.69) TNK2ALDH1A1CYP1A2MAPTCYP2C19
SCHEMBL1589145 0.69 HRH4 (0.68) TNK2ALDH1A1CYP1A2MAPTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105592850-A Inhibitors of ACK1/TNK2 tyrosine kinase H LEE MOFFITT CANCER CT &RES 2016-05-18 CN disclosed