SCHEMBL28068016

SCHEMBL28068016

O=[N+]([O-])c1cc2c(cnn2C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1I

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.35
PIN1 Q13526 2/20 0.34
HTT P42858 5/20 0.32
LMNA P02545 3/20 0.32
HPGD P15428 1/20 0.32
ATM Q13315 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GLS O94925 1/20 0.32
ALDH1A1 P00352 5/20 0.32
TDP1 Q9NUW8 2/20 0.31
MITF O75030 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PARP1 P09874 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28829273 0.85 LMNA (0.38) PIN1HTTLMNAHPGDATM
SCHEMBL16619910 0.85 CYP19A1 (0.34) HSP90AA1PIN1HTTLMNAHPGD
SCHEMBL18024520 0.83 ALDH1A1 (0.35) HSP90AA1PIN1HTTLMNAHPGD
SCHEMBL28067984 0.82 PIN1 (0.34) HSP90AA1PIN1HTTLMNAHPGD
SCHEMBL16619583 0.82 PIN1 (0.32) HSP90AA1PIN1HTTLMNAHPGD
SCHEMBL16619703 0.80 PIN1 (0.36) HSP90AA1PIN1GLSALDH1A1CYP1A2
SCHEMBL16619914 0.80 CYP1A2 (0.42) PIN1LMNAHPGDSMN1; SMN2ALDH1A1
SCHEMBL20475244 0.80 HSP90AA1 (0.32) HSP90AA1PIN1HTTLMNAHPGD
SCHEMBL29447518 0.78 MAPT (0.42) HTTLMNASMN1; SMN2GLSALDH1A1
SCHEMBL2279071 0.78 GLS (0.50) LMNASMN1; SMN2GLSALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105636586-A ERK inhibitors and methods of use ARAXES PHARMA LLC 2016-06-01 CN disclosed