SCHEMBL28068091

SCHEMBL28068091

COc1ccc(Cc2ccc3c(CC(=O)OCN)cn(S(=O)(=O)c4cccnc4)c3c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 10/20 0.42
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
PPARG P37231 2/20 0.38
PPARD Q03181 2/20 0.38
PPARA Q07869 2/20 0.38
CYP11B1 P15538 3/20 0.38
CYP11B2 P19099 3/20 0.38
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
KEAP1 Q14145 2/20 0.36
NFE2L2 Q16236 2/20 0.36
LMNA P02545 1/20 0.36
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR1E P28566 1/20 0.36
HTR1F P30939 1/20 0.36
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28068112 0.84 HTR6 (0.46) HTR6CHRNB4CHRNA3CYP11B1CYP11B2
SCHEMBL28068045 0.83 HTR6 (0.42) HTR6CHRNB4CHRNA3PPARGPPARD
Hydrochloric Acid SCHEMBL28068041 0.83 HTR6 (0.45) HTR6CHRNB4CHRNA3CYP11B1CYP11B2
SCHEMBL28068087 0.81 KMT2A (0.49) HTR6CHRNB4CHRNA3CYP11B1CYP11B2
SCHEMBL17971581 0.75 HTR6 (0.44) HTR6CYP2C9LMNAHTR1ADRD2
SCHEMBL19971359 0.75 HTR6 (0.42) HTR6CHRNB4CHRNA3PPARGPPARD
SCHEMBL16626785 0.74 HTR6 (0.44) HTR6CYP11B1CYP11B2HTR1ADRD2
SCHEMBL16626404 0.74 HTR6 (0.45) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL28829305 0.74 HTR6 (0.43) HTR6CHRNB4CHRNA3CYP2C9KEAP1
SCHEMBL16626784 0.74 HTR6 (0.42) HTR6PPARGPPARDPPARACYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612150-A Sulfonylindole derivatives and process for producing the same DAE WOONG PHARMA 2016-05-25 CN disclosed