SCHEMBL28068538

SCHEMBL28068538

O=C(O)C(Cl)c1ccccc1C1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C1 Q04828 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
GBA1 P04062 1/20 0.35
RBP4 P02753 2/20 0.35
HSD17B10 Q99714 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
NOTUM Q6P988 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP1A2 P05177 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C9 P11712 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10941871 0.83 PTGDR2 (0.34) PTGDR2AKR1C3AKR1C1HTTCYP2D6
SCHEMBL28068627 0.80 TSHR (0.39) ADRA2AADRA2BADRA2CGBA1MEN1
SCHEMBL21784784 0.79 MMP2 (0.42) PTGDR2ADRA2AADRA2BADRA2CGBA1
SCHEMBL14661272 0.78 PTGDR2 (0.47) PTGDR2
Ammonia Solution, Strong SCHEMBL28615660 0.75 ADRA2A (0.40) ADRA2AADRA2BADRA2CGBA1TSHR
SCHEMBL415803 0.74 PTGDR2 (0.45) PTGDR2ADRA2AKMT2ACYP1A2CYP2C9
SCHEMBL2062948 0.74 PTGDR2 (0.45) PTGDR2ADRA2AKMT2ACYP1A2CYP2C9
SCHEMBL418663 0.74 PTGDR2 (0.45) PTGDR2ADRA2AKMT2ACYP1A2CYP2C9
SCHEMBL198311 0.72 PTGDR2 (0.48) PTGDR2MEN1KMT2A
SCHEMBL198081 0.72 PTGDR2 (0.48) PTGDR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103687860-B As P2X7Heterocyclic amide derivatives of receptor antagonists 埃科特莱茵药品有限公司 2016-06-08 CN disclosed