SCHEMBL28068640

SCHEMBL28068640

COC(=O)Cc1ccc(Cl)cc1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
KDM4E B2RXH2 4/20 0.43
MAPT P10636 2/20 0.43
CYP1A2 P05177 1/20 0.43
GLA P06280 1/20 0.43
CYP3A4 P08684 1/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
F2 P00734 1/20 0.41
ALDH1A1 P00352 5/20 0.40
HTT P42858 4/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
ACLY P53396 1/20 0.39
THRB P10828 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
AKR1C3 P42330 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27033421 0.88 MAPT (0.46) HPGDNPSR1KDM4EMAPTCYP1A2
SCHEMBL29958664 0.88 MAPT (0.46) HPGDNPSR1KDM4EMAPTCYP1A2
SCHEMBL23599468 0.82 MAPT (0.43) HPGDNPSR1KDM4EMAPTCYP1A2
SCHEMBL18245557 0.82 KDM4E (0.43) HPGDKDM4EMAPTCYP1A2GLA
SCHEMBL2437800 0.82 NPC1 (0.55) HPGDKDM4EMAPTCYP1A2GLA
SCHEMBL4689558 0.80 ADRA1D (0.43) HPGDNPSR1F2ALDH1A1MEN1
SCHEMBL837451 0.79 ALDH1A1 (0.56) KDM4EMAPTGAAALDH1A1HTT
SCHEMBL1525623 0.78 ALDH1A1 (0.54) KDM4EMAPTGAAALDH1A1HTT
SCHEMBL20521859 0.78 MEN1 (0.47) HPGDKDM4EMAPTGLAGAA
SCHEMBL10923842 0.78 ALDH1A1 (0.50) KDM4EMAPTCYP1A2CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103687860-B As P2X7Heterocyclic amide derivatives of receptor antagonists 埃科特莱茵药品有限公司 2016-06-08 CN disclosed