SCHEMBL28068816

SCHEMBL28068816

C[C@@H]1CN(CC(=N)NO)CCN1C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.33
TSHR P16473 1/20 0.33
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
MGLL Q99685 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16400400 1.00 SIGMAR1 (0.33) SIGMAR1TSHRDRD2DRD3MGLL
SCHEMBL17867679 0.81 SETD7 (0.37) TSHRSMN1; SMN2
SCHEMBL17867678 0.81 SETD7 (0.37) TSHRSMN1; SMN2
SCHEMBL13733481 0.80 HSD17B10 (0.37) SIGMAR1TSHRDRD2DRD3MGLL
SCHEMBL13733486 0.80 HSD17B10 (0.37) SIGMAR1TSHRDRD2DRD3MGLL
SCHEMBL16400765 0.78 GBA2 (0.37) SIGMAR1TSHRDRD2DRD3SMN1; SMN2
SCHEMBL18691907 0.73 HSD11B1 (0.43) SIGMAR1DRD2DRD3SMN1; SMN2
SCHEMBL13662624 0.72 P2RX7 (0.42) DRD2DRD3PTGDR2SMN1; SMN2
SCHEMBL21772146 0.72 MAPK1 (0.50) TSHRDRD2DRD3MGLLPTGDR2
SCHEMBL22117940 0.72 MAPK1 (0.50) TSHRDRD2DRD3MGLLPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555783-B Include the autotaxin inhibitors of heteroaromatic rings benzyl amide ring core 诺华股份有限公司 2017-12-01 CN disclosed
CN-105555783-A Autotaxin inhibitors comprising a heteroaromatic ring-benzyl-amide-cycle core NOVARTIS AG 2016-05-04 CN disclosed