SCHEMBL28070637

SCHEMBL28070637

COc1ccc(-c2n[nH]nc2C)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
XDH P47989 2/20 0.47
ALDH1A1 P00352 4/20 0.46
HPGD P15428 2/20 0.46
PTGS2 P35354 1/20 0.46
ATM Q13315 1/20 0.45
KDM4E B2RXH2 3/20 0.44
LMNA P02545 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
GAA P10253 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17584763 0.88 MEN1 (0.59) MEN1KMT2AXDHALDH1A1HPGD
SCHEMBL17141308 0.79 MEN1 (0.51) MEN1KMT2AXDHALDH1A1KDM4E
SCHEMBL10166458 0.75 ALOX15 (0.70) ALDH1A1HPGDPTGS2ATMKDM4E
SCHEMBL10508211 0.75 ALDH1A1 (0.60) MEN1KMT2AALDH1A1HPGDPTGS2
SCHEMBL31438211 0.75 ERBB2 (0.68) MEN1KMT2AXDHALDH1A1HPGD
SCHEMBL408607 0.74 TGFBR1 (0.56) MEN1KMT2AALDH1A1HPGDATM
SCHEMBL17141287 0.74 TUBB4A (0.57) MEN1KMT2ALMNAMAPT
SCHEMBL10814624 0.74 MEN1 (0.77) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL28058395 0.74 MAPK8 (0.49) LMNATDP1MAPT
SCHEMBL5223142 0.73 MEN1 (0.53) MEN1KMT2AXDHALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105669569-B A kind of synthetic method of the triazole compounds of NH 1,2,3 武汉工程大学 2017-12-12 CN disclosed
CN-105669569-A Synthesis method of NH-1,2,3-triazole compound 武汉工程大学 2016-06-15 CN disclosed