SCHEMBL28072772

SCHEMBL28072772

COC(=O)c1ccc(C(Cl)C(N)=O)c([N+](=O)[O-])c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.53
PDK1 Q15118 1/20 0.51
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
LMNA P02545 2/20 0.47
KMT2A Q03164 2/20 0.46
PKM P14618 1/20 0.46
MAPT P10636 3/20 0.44
HSP90AA1 P07900 1/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 2/20 0.44
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8474404 0.82 PDK1 (0.65) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL351791 0.81 VCAM1 (0.50) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL4122879 0.81 VCAM1 (0.58) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL18148190 0.80 VCAM1 (0.57) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL30635851 0.80 ALDH1A1 (0.62) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL12138038 0.80 ALDH1A1 (0.62) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL21932200 0.78 VCAM1 (0.56) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL2949996 0.77 VCAM1 (0.54) VCAM1PDK1ALDH1A1HPGDNPSR1
SCHEMBL5734347 0.77 VCAM1 (0.68) VCAM1ALDH1A1HPGDNPSR1LMNA
SCHEMBL28548226 0.76 VCAM1 (0.53) VCAM1PDK1ALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104016927-B Pyrimidine mercaptoacetamide derivative and preparation method thereof and application 山东大学 2016-06-22 CN disclosed