SCHEMBL28073005

SCHEMBL28073005

CC(C)S(=O)(=O)c1ccc(C#N)cc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 3/20 0.40
RAD51 Q06609 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
XDH P47989 1/20 0.36
ATR Q13535 2/20 0.36
BRPF1 P55201 2/20 0.35
GRIA4 P48058 2/20 0.35
GRIA1 P42261 1/20 0.35
GRIA2 P42262 1/20 0.35
GRIA3 P42263 1/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35
EPAS1 Q99814 1/20 0.34
CASP3 P42574 1/20 0.34
HSD11B1 P28845 1/20 0.34
BRD1 O95696 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18229960 0.81 TRPV4 (0.43) TRPV4RAD51KDM4EALDH1A1GAA
SCHEMBL21773502 0.80 HSD11B1 (0.48) TRPV4HSD11B1
SCHEMBL3782276 0.79 CA1 (0.47) TRPV4RAD51KDM4EALDH1A1GAA
SCHEMBL16676516 0.78 TRPV4 (0.48) TRPV4RAD51KDM4EALDH1A1GAA
SCHEMBL6405238 0.76 XDH (0.37) KDM4EALDH1A1GAAXDH
SCHEMBL10127000 0.75 TDP1 (0.45) KDM4EALDH1A1CA1
SCHEMBL123288 0.74 RAD51 (0.49) TRPV4RAD51GRIA4GRIA1GRIA2
SCHEMBL14866077 0.74 CYP3A4 (0.44) TRPV4KDM4EALDH1A1GAACA1
SCHEMBL20085640 0.74 NPC1 (0.42) ALDH1A1
SCHEMBL12491217 0.74 CA2 (0.39) KDM4ECA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829285-A Quinazolinone and isoquinolinone derivatives 中外制药株式会社 2016-08-03 CN disclosed