SCHEMBL28073015

SCHEMBL28073015

CCSc1ccc(Br)cc1NC

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.36
DDR1 Q08345 3/20 0.35
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CCR2 P41597 2/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
ADRA2A P08913 2/20 0.31
ADRA2B P18089 2/20 0.31
ADRA2C P18825 2/20 0.31
ADRA1D P25100 2/20 0.31
ADRA1A P35348 2/20 0.31
ADRA1B P35368 2/20 0.31
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16676458 0.84 MAPT (0.36) DDR1MAPTSMN1; SMN2CCR2ADRA2A
SCHEMBL27999924 0.79 CCR2 (0.47) DDR1SMN1; SMN2CCR2ADRA2AADRA2B
SCHEMBL25456570 0.79 CCR2 (0.43) HDAC6MAPTSMN1; SMN2CCR2
Hydrochloric Acid SCHEMBL28000103 0.78 CCR2 (0.46) DDR1SMN1; SMN2CCR2ADRA2AADRA2B
SCHEMBL25872926 0.78 DDR1 (0.46) HDAC6DDR1MAPTSMN1; SMN2CCR2
SCHEMBL28072988 0.75 CYP1A2 (0.41) MAPTSMN1; SMN2ADRA2AADRA2CADRA1D
SCHEMBL28000085 0.75 AOC3 (0.36) HDAC6CCR2
SCHEMBL25302556 0.75 PKM (0.43) DDR1MAPTSMN1; SMN2
SCHEMBL25924438 0.74 CHRNB2 (0.30) CHRNB2CHRNA7CHRNA4
SCHEMBL2416681 0.73 TSHR (0.36) DDR1MAPTSMN1; SMN2CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829285-A Quinazolinone and isoquinolinone derivatives 中外制药株式会社 2016-08-03 CN disclosed