SCHEMBL16664909

SCHEMBL16664909

CCCNc1cc(-c2cnc(C(F)(F)F)nc2)ncn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.43
TSHR P16473 5/20 0.43
CYP2C19 P33261 5/20 0.43
CYP3A4 P08684 4/20 0.43
ALOX15 P16050 3/20 0.43
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
FAAH O00519 5/20 0.39
CYP2D6 P10635 4/20 0.37
HIF1A Q16665 2/20 0.37
CYP2C9 P11712 1/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MAPK1 P28482 1/20 0.37
FLT3 P36888 1/20 0.37
TYRO3 Q06418 1/20 0.37
MERTK Q12866 1/20 0.37
GAS6 Q14393 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16664911 0.85 FAAH (0.43) CYP1A2TSHRCYP2C19CYP3A4ALOX15
SCHEMBL16664949 0.85 FLT3 (0.39) CYP1A2TSHRCYP2C19CYP3A4ALOX15
SCHEMBL28074525 0.81 CYP1A2 (0.52) CYP1A2TSHRCYP2C19CYP3A4ALOX15
SCHEMBL16664979 0.79 FAAH (0.39) CYP1A2TSHRCYP2C19CYP3A4ALOX15
SCHEMBL16665010 0.79 FAAH (0.41) CYP1A2CYP2C19CYP3A4HSD17B10KDM4E
SCHEMBL18627048 0.77 ABL1 (0.44) CYP1A2TSHRCYP2C19CYP3A4ALOX15
SCHEMBL16664919 0.75 PIK3CA (0.44) CYP1A2CYP2C19CYP3A4ALOX15HSD17B10
SCHEMBL15343048 0.75 KDM4E (0.47) CYP1A2CYP2C19CYP3A4HSD17B10KDM4E
SCHEMBL16664969 0.75 KDM4E (0.47) CYP1A2CYP2C19CYP3A4HSD17B10KDM4E
SCHEMBL18902711 0.75 CYP1A2 (0.53) CYP1A2TSHRCYP2C19CYP3A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058031-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2015-04-23 WO disclosed