SCHEMBL28074646

SCHEMBL28074646

CNc1ccnc(-c2cnc(C(F)(F)F)nc2)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.36
TRPV3 Q8NET8 1/20 0.36
KIF11 P52732 1/20 0.35
KDM4E B2RXH2 1/20 0.34
TGFBR1 P36897 1/20 0.34
MAPKAPK2 P49137 2/20 0.33
ABL1 P00519 3/20 0.33
IDH1 O75874 1/20 0.33
HDAC1 Q13547 1/20 0.33
PTGES O14684 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE11A Q9HCR9 1/20 0.32
PRKCA P17252 1/20 0.32
BCR P11274 2/20 0.32
PLK1 P53350 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16894177 0.82 ABL1 (0.43) TRPV3KDM4ETGFBR1ABL1BCR
SCHEMBL25755088 0.79 KIF11 (0.56) TRPV3KIF11TGFBR1MAPKAPK2ABL1
SCHEMBL20224615 0.79 CCR1 (0.53) TRPA1TRPV3KDM4EABL1BCR
SCHEMBL20224620 0.77 RAD51 (0.41) TRPA1TRPV3KDM4ETGFBR1HDAC1
SCHEMBL20224616 0.77 NOS3 (0.47) KIF11TGFBR1ABL1HDAC1BCR
SCHEMBL20224612 0.76 NOS3 (0.36) TRPA1TRPV3KIF11TGFBR1HDAC1
SCHEMBL30636782 0.75 CCR1 (0.48) KDM4ETGFBR1MAPKAPK2PRKCAPLK1
SCHEMBL2521580 0.75 CCR1 (0.48) KDM4ETGFBR1MAPKAPK2PRKCAPLK1
SCHEMBL21022111 0.73 TGFBR1 (0.48) KDM4ETGFBR1MAPKAPK2
SCHEMBL17039389 0.73 KIF11 (0.39) TRPV3KIF11PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed