SCHEMBL28074688

SCHEMBL28074688

CN1C(=O)C(=O)c2c(N)cccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.50
CES1 P23141 1/20 0.50
ADORA2A P29274 3/20 0.41
PTPRC P08575 1/20 0.41
DPP4 P27487 1/20 0.41
HSPA1A P0DMV8 1/20 0.40
PABPC1 P11940 1/20 0.40
ADRA2C P18825 1/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
ATM Q13315 2/20 0.39
USP2 O75604 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
CASP3 P42574 2/20 0.38
THRB P10828 1/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
FGR P09769 1/20 0.36
PIM1 P11309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7756746 0.82 TTR (0.52) TTRCES1DPP4KMT2AMEN1
SCHEMBL21848273 0.77 TTR (0.50) TTRCES1KMT2AMEN1CASP3
SCHEMBL1137933 0.77 TTR (0.55) TTRCES1DPP4KMT2AMEN1
SCHEMBL15206754 0.77 TTR (0.50) TTRCES1KMT2AMEN1CASP3
SCHEMBL754994 0.77 CES1 (0.50) TTRCES1KMT2AMEN1CASP3
SCHEMBL2290914 0.77 TTR (0.50) TTRCES1KMT2AMEN1CASP3
SCHEMBL14880102 0.77 MEN1 (0.46) TTRCES1DPP4KMT2AMEN1
SCHEMBL9728201 0.77 ALDH1A1 (0.48) CES1ADORA2APTPRCDPP4PABPC1
SCHEMBL28074698 0.76 TTR (0.48) TTRCES1DPP4KMT2AMEN1
SCHEMBL30067921 0.74 TTR (0.47) TTRCES1KMT2AMEN1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105732476-B A kind of carbazole isatin type compound and its preparation method and purposes 吉首大学 2017-12-01 CN disclosed
CN-105732476-A Carbazole-isatin type compound and preparation method and application thereof 吉首大学 2016-07-06 CN disclosed