SCHEMBL2807618

SCHEMBL2807618

Cc1cc(N)cc(C#CC(C)(C)O)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
TSHR P16473 1/20 0.44
PAK4 O96013 3/20 0.35
PAK1 Q13153 1/20 0.35
PKN1 Q16512 1/20 0.35
ASIC3 Q9UHC3 1/20 0.34
PIKFYVE Q9Y2I7 4/20 0.33
TTBK1 Q5TCY1 3/20 0.33
MAP3K14 Q99558 3/20 0.32
FFAR1 O14842 1/20 0.32
PTGES2 Q9H7Z7 2/20 0.31
HAO1 Q9UJM8 2/20 0.31
KDM4E B2RXH2 1/20 0.31
KMT2A Q03164 1/20 0.30
ATM Q13315 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25061870 0.78 ASIC3 (0.34) PAK4PAK1PKN1ASIC3MAP3K14
SCHEMBL30092382 0.74 MAP3K14 (0.45) ALDH1A1PAK4PAK1PKN1ASIC3
SCHEMBL471131 0.74 MAP3K14 (0.45) ALDH1A1PAK4PAK1PKN1ASIC3
SCHEMBL3570374 0.73 CHRNB2 (0.42) ALDH1A1PAK4PAK1PKN1ASIC3
SCHEMBL3448180 0.72 APP (0.54) TSHRPAK4PAK1PKN1ASIC3
SCHEMBL2629434 0.72 GRM5 (0.49) ASIC3MAP3K14FFAR1HAO1
SCHEMBL14268091 0.70 ASIC3 (0.49) ALDH1A1TSHRASIC3FFAR1PTGES2
SCHEMBL19720165 0.70 GABRA1 (0.36) ALDH1A1TSHRPAK4PAK1PKN1
SCHEMBL1466752 0.69 PAK4 (0.42) ALDH1A1PAK4PAK1PKN1ASIC3
SCHEMBL13692781 0.68 ASIC3 (0.34) TSHRPAK4PAK1PKN1ASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B ALDH1A1 401/4885TSHR 3644/4885PAK4 4788/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 ALDH1A1 1480/4885TSHR 4692/4885PAK4 4405/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.