SCHEMBL28076875

SCHEMBL28076875

Cc1c(-c2ccc(CN)cc2)ccc2c1OC(C)(C)C2

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.42
AKT2 P31751 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
POLB P06746 1/20 0.34
LMNA P02545 2/20 0.33
HTR1A P08908 1/20 0.33
HTR2A P28223 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 2/20 0.32
TAAR1 Q96RJ0 1/20 0.32
DHFR P00374 1/20 0.32
PDCD1 Q15116 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28076657 0.76 HTR2A (0.38) CD274FFAR4HRH3HTR2ADHFR
SCHEMBL28076877 0.72 HRH3 (0.42) CD274HRH3HTR2ATAAR1
SCHEMBL28076654 0.70 CD274 (0.40) CD274AKT2FFAR4HRH3NPC1
SCHEMBL657575 0.70 ALDH1A1 (0.46) SMN1; SMN2POLBLMNAHTR1AALDH1A1
SCHEMBL112586 0.68 LMNA (0.44) NPC1POLBLMNAALDH1A1KDM4E
SCHEMBL22866559 0.66 CD274 (0.61) CD274AKT2HRH3TAAR1PDCD1
SCHEMBL25570163 0.66 HTR2A (0.42) FFAR4HTR2ADHFR
SCHEMBL13156334 0.65 HIF1A (0.44) HTR2AALDH1A1KDM4E
SCHEMBL8123158 0.64 DHFR (0.37) SMN1; SMN2POLBLMNAHTR2AALDH1A1
SCHEMBL435089 0.63 LMNA (0.49) NPC1SMN1; SMN2POLBLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965147-B Benzofuran derivatives 武田药品工业株式会社 2016-08-24 CN disclosed