SCHEMBL28077039

SCHEMBL28077039

C=C(c1cc(F)ccc1F)C(C)C#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.43
CES1 P23141 3/20 0.43
CA3 P07451 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
PSMB11 A5LHX3 1/20 0.33
PSMA7 O14818 1/20 0.33
PSMB1 P20618 1/20 0.33
PSMA1 P25786 1/20 0.33
PSMA2 P25787 1/20 0.33
PSMA3 P25788 1/20 0.33
PSMA4 P25789 1/20 0.33
PSMB8 P28062 1/20 0.33
PSMB9 P28065 1/20 0.33
PSMA5 P28066 1/20 0.33
PSMB4 P28070 1/20 0.33
PSMB6 P28072 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12909551 0.80 CES2 (0.50) CES2CES1CA3CA6CA5A
SCHEMBL1012686 0.79 CES2 (0.48) CES2CES1CA3CA6CA5A
SCHEMBL1012685 0.79 CES2 (0.48) CES2CES1CA3CA6CA5A
SCHEMBL11042341 0.70 CES2 (0.56) CES2CES1CA3CA6CA5A
SCHEMBL28319857 0.70 CES2 (0.53) CES2CES1
SCHEMBL16510004 0.69 CES2 (0.39) CES2CES1CA3CA6CA5A
SCHEMBL12289224 0.66 CES2 (0.56) CES2CES1CA3CA6CA5A
SCHEMBL31504503 0.66 PSEN1 (0.42) CES2CES1CA3CA6CA5A
SCHEMBL12909549 0.66 CES2 (0.61) CES2CES1CA3CA6CA5A
SCHEMBL3632173 0.66 CES2 (0.46) CES2CES1CA3CA6CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105732605-A Preparation method of isavuconazole intermediate 山东亨利医药科技有限责任公司 2016-07-06 CN claimed
CN-105732605-A Preparation method of isavuconazole intermediate 山东亨利医药科技有限责任公司 2016-07-06 CN disclosed