SCHEMBL28077290

SCHEMBL28077290

NS(=O)(=O)c1ccc(Nc2ccc3ccncc3c2)cc1.[H+]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 13/20 0.50
CA2 P00918 13/20 0.50
CA9 Q16790 13/20 0.50
CA12 O43570 8/20 0.50
SOS1 Q07889 3/20 0.50
CA14 Q9ULX7 4/20 0.49
CA6 P23280 3/20 0.49
CA7 P43166 3/20 0.49
CA4 P22748 2/20 0.49
CA13 Q8N1Q1 2/20 0.49
CA5A P35218 2/20 0.49
DKK1 O94907 1/20 0.48
GSK3B P49841 1/20 0.48
CDK2 P24941 1/20 0.48
KDR P35968 1/20 0.47
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
KMT2A Q03164 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
ROCK1 Q13464 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550093 0.85 LMNA (0.58) CA1CA2CA9CA12CA14
SCHEMBL28746782 0.79 LMNA (0.70) CA1CA2CA9CA12SOS1
SCHEMBL566973 0.78 LMNA (0.58) CA1CA2CA9CA12MEN1
SCHEMBL31203257 0.78 LMNA (0.58) CA1CA2CA9CA12MEN1
SCHEMBL12278421 0.78 SOS1 (0.58) CA1CA2CA9CA12SOS1
Hydrochloric Acid SCHEMBL22129912 0.77 LMNA (0.56) CA1CA2CA9CA12MEN1
SCHEMBL18311786 0.77 ALDH1A1 (0.63) MEN1KMT2AROCK1
SCHEMBL24125025 0.75 IMPDH2 (0.45)
SCHEMBL27823663 0.74 CA2 (0.58) CA1CA2CA9CA12SOS1
SCHEMBL28107398 0.74 SOS1 (0.70) CA1CA2CA9CA12SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105764510-A An H3 receptor antagonist combined with a cholinesterase inhibitor for use in the treatment of alzheimer's disease 赛诺菲 2016-07-13 CN disclosed