SCHEMBL28078713

SCHEMBL28078713

NC(=O)c1cccc(-c2cccc(S(N)(=O)=O)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.54
CA1 P00915 7/20 0.54
CA9 Q16790 7/20 0.54
CA12 O43570 6/20 0.54
ERN1 O75460 2/20 0.53
IKBKB O14920 1/20 0.52
CA14 Q9ULX7 2/20 0.51
PTGES2 Q9H7Z7 1/20 0.49
ADAMTS4 O75173 1/20 0.48
GAA P10253 1/20 0.48
PARP1 P09874 1/20 0.47
CA4 P22748 1/20 0.47
CDK8 P49336 1/20 0.47
CA13 Q8N1Q1 1/20 0.46
DHODH Q02127 1/20 0.46
NOS1 P29475 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1805285 0.89 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL30230622 0.89 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL30903622 0.88 CA2 (0.69) CA2CA1CA9CA12ERN1
SCHEMBL3720556 0.88 CA2 (0.69) CA2CA1CA9CA12ERN1
SCHEMBL3655412 0.85 CAMKK2 (0.55) CA2CA1CA9CA12ERN1
SCHEMBL31422694 0.83 PARP1 (0.64) ERN1PARP1CDK8DHODH
SCHEMBL2431097 0.83 PARP1 (0.64) ERN1PARP1CDK8DHODH
SCHEMBL6999225 0.81 DHODH (0.63) ERN1PARP1CDK8DHODH
SCHEMBL28032548 0.81 CA2 (0.73) CA2CA1CA9CA12CA14
SCHEMBL13742952 0.81 CA12 (0.81) CA2CA1CA9CA12ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683157-B Sulfonamides as sodium channel modulators 沃泰克斯药物股份有限公司 2019-07-19 CN disclosed
CN-105683157-A Sulfonamides as modulators of sodium channels 沃泰克斯药物股份有限公司 2016-06-15 CN disclosed