Pirfenidone

Pirfenidone

SCHEMBL28079090

Cc1ccc(=O)n(-c2ccccc2)c1.[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.96
ALDH1A1 P00352 3/20 0.96
CYP1A2 P05177 2/20 0.96
HPGD P15428 1/20 0.96
BLM P54132 1/20 0.96
HSD17B10 Q99714 1/20 0.96
MAPK14 Q16539 5/20 0.48
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 2/20 0.42
POLB P06746 1/20 0.42
COMT P21964 1/20 0.41
NAPRT Q6XQN6 1/20 0.39
FGFR1 P11362 1/20 0.39
CA12 O43570 1/20 0.38
BRD4 O60885 1/20 0.38
BRPF1 P55201 1/20 0.38
CA9 Q16790 1/20 0.38
KAT2B Q92831 1/20 0.38
BRD9 Q9H8M2 1/20 0.38
NOTUM Q6P988 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pirfenidone SCHEMBL4708 0.98 KDM4E (1.00) KDM4EALDH1A1CYP1A2HPGDBLM
Pirfenidone SCHEMBL1006039 0.98 KDM4E (1.00) KDM4EALDH1A1CYP1A2HPGDBLM
Pirfenidone SCHEMBL22492268 0.96 KDM4E (0.96) KDM4EALDH1A1CYP1A2HPGDBLM
Pirfenidone SCHEMBL28532042 0.96 KDM4E (0.96) KDM4EALDH1A1CYP1A2HPGDBLM
Pirfenidone SCHEMBL28115013 0.89 KDM4E (0.83) KDM4EALDH1A1CYP1A2HPGDBLM
Pirfenidone SCHEMBL27872362 0.89 ALDH1A1 (0.83) KDM4EALDH1A1CYP1A2HPGDBLM
SCHEMBL356681 0.87 ALDH1A1 (0.80) KDM4EALDH1A1CYP1A2HPGDBLM
SCHEMBL10059357 0.87 KDM4E (0.79) KDM4EALDH1A1CYP1A2HPGDBLM
SCHEMBL3970272 0.85 ALDH1A1 (0.77) KDM4EALDH1A1CYP1A2HPGDBLM
Deupirfenidone SCHEMBL4059454 0.85 KDM4E (0.76) KDM4EALDH1A1CYP1A2HPGDBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112912386-A Cell penetrating peptide based on influenza virus M2 protein 中国医学科学院基础医学研究所 2021-06-04 CN claimed
CN-109010916-B Moldable formulations containing oxysterol in acellular tissue matrices 华沙整形外科股份有限公司 2022-03-04 CN disclosed
CN-108786619-B Bone material dispensing apparatus and method 华沙整形外科股份有限公司 2022-03-04 CN disclosed
CN-105517557-B Bacterial strains having antimicrobial activity and biocontrol compositions comprising said strains 特雷根控股有限公司 2021-11-30 CN disclosed
CN-110655585-A Synthetic polypeptides and uses thereof 中央研究院 2020-01-07 CN disclosed
CN-105793255-A Heterocyclic compounds and their use 无限药品股份有限公司 2016-07-20 CN disclosed