SCHEMBL28079205

SCHEMBL28079205

O=CNc1n[nH]c2ccc(CN3CCCC3)cc12

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 13/20 0.48
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
INSR P06213 1/20 0.44
IGF1R P08069 1/20 0.44
ALK Q9UM73 1/20 0.44
WNT1 P04628 4/20 0.43
DYRK1A Q13627 4/20 0.43
CLK2 P49760 2/20 0.43
CLK3 P49761 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11748510 0.79 NTRK1 (0.43) KDM4EALDH1A1
SCHEMBL28079288 0.79 NTRK1 (0.45) MCHR1
SCHEMBL1966636 0.74 DYRK1A (0.55) CDK5CDK5R1WNT1DYRK1ACLK2
SCHEMBL28079206 0.73 DYRK1A (0.69) CDK5CDK5R1WNT1DYRK1ACLK2
SCHEMBL25200397 0.71 PDPK1 (0.53) CDK5ALKDYRK1ACLK2
SCHEMBL3513100 0.71 ALK (0.73) INSRIGF1RALKCLK2
SCHEMBL3514493 0.70 ALK (0.74) INSRIGF1RALKCLK2
SCHEMBL26393980 0.68 GSK3B (0.57) DYRK1A
SCHEMBL11748390 0.68 FADS1 (0.54) KDM4E
SCHEMBL11754096 0.67 TRPA1 (0.50) KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658640-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed