SCHEMBL28079206

SCHEMBL28079206

NC(=O)c1n[nH]c2ccc(CN3CCCC3)cc12

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 19/20 0.69
WNT1 P04628 9/20 0.69
CLK2 P49760 5/20 0.69
CLK3 P49761 5/20 0.69
CDK5 Q00535 1/20 0.54
CDK5R1 Q15078 1/20 0.54
GSK3B P49841 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1966636 0.88 DYRK1A (0.55) DYRK1AWNT1CLK2CLK3CDK5
SCHEMBL17096993 0.83 DYRK1A (0.98) DYRK1AWNT1CLK2CLK3
SCHEMBL17095632 0.82 DYRK1A (1.00) DYRK1AWNT1CLK2CLK3
SCHEMBL17096954 0.82 DYRK1A (1.00) DYRK1AWNT1CLK2CLK3
SCHEMBL7532630 0.81 JAK2 (0.55) DYRK1AWNT1CLK2CLK3GSK3B
SCHEMBL17096358 0.81 DYRK1A (0.94) DYRK1AWNT1CLK2CLK3
SCHEMBL17096641 0.80 DYRK1A (0.73) DYRK1AWNT1CLK2CLK3GSK3B
SCHEMBL28079290 0.79 PRKAG1 (0.48) DYRK1AWNT1CLK2CLK3GSK3B
SCHEMBL13554360 0.78 JAK2 (0.50) DYRK1AWNT1CLK2CLK3GSK3B
SCHEMBL28087969 0.77 CLK2 (0.47) DYRK1AWNT1CLK2CLK3CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658640-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed