SCHEMBL28087969

SCHEMBL28087969

NC(=O)c1n[nH]c2ccc(CC34CCN(CC3)CC4)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK2 P49760 4/20 0.47
CLK3 P49761 4/20 0.47
DYRK1A Q13627 4/20 0.47
WNT1 P04628 3/20 0.47
GSK3B P49841 2/20 0.38
ACACB O00763 1/20 0.38
ACACA Q13085 1/20 0.38
NTRK1 P04629 3/20 0.38
LRRK2 Q5S007 1/20 0.37
MAP4K4 O95819 1/20 0.36
FLT3 P36888 1/20 0.36
HAO1 Q9UJM8 1/20 0.36
DDR1 Q08345 1/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
JAK3 P52333 1/20 0.35
PRKAB2 O43741 2/20 0.35
PRKAG1 P54619 2/20 0.35
PRKAA2 P54646 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28079206 0.77 DYRK1A (0.69) CLK2CLK3DYRK1AWNT1GSK3B
SCHEMBL28079290 0.76 PRKAG1 (0.48) CLK2CLK3DYRK1AWNT1GSK3B
SCHEMBL13554360 0.75 JAK2 (0.50) CLK2CLK3DYRK1AWNT1GSK3B
SCHEMBL8877161 0.72 JAK2 (0.54) CLK2CLK3DYRK1AWNT1NTRK1
SCHEMBL12339927 0.71 GSK3B (0.49) CLK2CLK3DYRK1AWNT1GSK3B
SCHEMBL3603302 0.71 WNT1 (0.40) CLK2CLK3DYRK1AWNT1ACACB
SCHEMBL28258471 0.70 NTRK1 (0.43) CLK2CLK3DYRK1AWNT1GSK3B
SCHEMBL23368472 0.70 GSK3B (0.47) CLK2CLK3DYRK1AWNT1GSK3B
Hydrochloric Acid SCHEMBL27980243 0.69 ULK1 (0.45) CLK2CLK3DYRK1AWNT1GSK3B
SCHEMBL591164 0.69 HTR1A (0.48) CLK2CLK3DYRK1AWNT1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104193741-B Quinuclidine-4-ylmethyl 1H-indole-3-carboxylic acid ester derivant as alpha 7 nicotinic acetylcholine receptor ligands 阿尔法梅根有限责任公司 2016-08-24 CN disclosed