SCHEMBL28079734

SCHEMBL28079734

CCc1ccc(-c2ccc(Cl)cc2)cc1C1=C(S(C)(=O)=O)C(C)=NN(C)C1C(=O)C1C(c2cc(-c3ccc(Cl)cc3)ccc2CC)=C(S(C)(=O)=O)C(C)=NN1C

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.35
CHRNA7 P36544 3/20 0.32
PTGS1 P23219 1/20 0.32
BRD4 O60885 1/20 0.32
NR1H2 P55055 2/20 0.32
MALT1 Q9UDY8 1/20 0.32
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
MAP4K4 O95819 1/20 0.31
RXRA P19793 1/20 0.31
NR1H3 Q13133 1/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL469885 0.65 BRD4 (0.37) BRD4
SCHEMBL470078 0.60 NPC1 (0.36) BRD4
SCHEMBL15086668 0.60 NPC1 (0.37) BRD4
SCHEMBL12603786 0.59 ALOX5 (0.41) RXRA
SCHEMBL15086669 0.59 NPC1 (0.41)
SCHEMBL12603775 0.58 AHR (0.50)
Acetic Acid SCHEMBL452190 0.57 HSD17B1 (0.40)
SCHEMBL469883 0.57 NPC1 (0.35)
SCHEMBL468935 0.57 ACACB (0.36)
SCHEMBL559918 0.57 ALDH1A1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104326952-B Prepare method and its intermediate of pyridazinone compound 住友化学株式会社 2016-08-24 CN disclosed