SCHEMBL28517969

SCHEMBL28517969

CNc1cn(Cc2cc(F)c(OC)c(F)c2)nn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.40
CACNA1H O95180 4/20 0.40
CACNA1G O43497 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
DBH P09172 1/20 0.40
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 2/20 0.38
HDAC1 Q13547 1/20 0.36
KCNH2 Q12809 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35
TUBA1A Q71U36 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28523893 0.85 SIGMAR1 (0.43) SIGMAR1HSP90AA1HSP90AB1KCNH2
SCHEMBL21491970 0.78 CYP19A1 (0.41) CACNA1HCACNA1GCACNA1IDBHHSP90AA1
SCHEMBL19611853 0.77 MEN1 (0.56) HSP90AA1HSP90AB1HDAC1MEN1KMT2A
SCHEMBL28080410 0.75 SIGMAR1 (0.56) SIGMAR1HDAC1KCNH2
Hydrochloric Acid SCHEMBL28523889 0.74 TAS2R8 (0.42) CACNA1HCACNA1GCACNA1IDBHKCNH2
SCHEMBL28525714 0.72 CACNA1H (0.40) CACNA1HCACNA1GCACNA1IDBH
SCHEMBL27971447 0.71 SIGMAR1 (0.59) SIGMAR1NPC1RAB9A
SCHEMBL9369847 0.71 CA5A (0.54) SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL21492020 0.67 DBH (0.40) CACNA1HCACNA1GCACNA1IDBHKCNH2
SCHEMBL17316286 0.66 L3MBTL1 (0.55) CACNA1HCACNA1GCACNA1IDBHMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed
CN-112218865-A Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2021-01-12 CN disclosed