SCHEMBL28080600

SCHEMBL28080600

N#CCC(=O)Nc1ccc(-c2ncnc3[nH]ccc23)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CIT O14578 1/20 0.58
JAK3 P52333 8/20 0.55
IKBKB O14920 1/20 0.53
CHUK O15111 1/20 0.53
JAK1 P23458 5/20 0.53
JAK2 O60674 6/20 0.50
HDAC6 Q9UBN7 3/20 0.49
ROCK2 O75116 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP3A5 P20815 1/20 0.49
LIMK1 P53667 1/20 0.49
BTK Q06187 2/20 0.49
MELK Q14680 2/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
PDGFRB P09619 1/20 0.46
KIT P10721 1/20 0.46
FLT3 P36888 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28080559 0.86 JAK3 (0.74) JAK3JAK1JAK2ROCK2CYP3A4
SCHEMBL30009846 0.81 CIT (0.65) CITJAK1
SCHEMBL28871098 0.81 CIT (0.63) CITJAK3IKBKBCHUKJAK1
SCHEMBL30009442 0.77 CIT (0.62) CITJAK3IKBKBCHUKJAK1
SCHEMBL30009111 0.77 ROCK2 (0.60) CITJAK3IKBKBCHUKJAK1
SCHEMBL28345572 0.77 JAK3 (0.74) CITJAK3IKBKBCHUKJAK1
SCHEMBL27387789 0.76 BTK (0.65) CITJAK3IKBKBCHUKJAK1
SCHEMBL29291567 0.76 CIT (0.57) CITJAK3IKBKBCHUKJAK1
SCHEMBL101362 0.74 JAK2 (0.53) CITJAK3IKBKBJAK1JAK2
SCHEMBL30009301 0.74 JAK1 (0.59) CITJAK3IKBKBCHUKJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712998-B Azaindole derivatives, preparation method and medical application thereof 上海润诺生物科技有限公司 2019-12-13 CN disclosed
CN-105712998-A Azaindole derivatives, preparation method and applications thereof in medicine 上海润诺生物科技有限公司 2016-06-29 CN disclosed