SCHEMBL2808160

SCHEMBL2808160

CC(O)COC(=O)/C=C/C(=O)OCC(C)O

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
MAPT P10636 2/20 0.44
HCAR2 Q8TDS4 7/20 0.43
ATM Q13315 1/20 0.43
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4444141 1.00 TSHR (0.52) TSHRMAPTHCAR2ATMKEAP1
SCHEMBL2465097 1.00 TSHR (0.52) TSHRMAPTHCAR2ATMKEAP1
SCHEMBL8640652 0.91 HCAR2 (0.54) TSHRMAPTHCAR2ATMKEAP1
SCHEMBL8639051 0.91 HCAR2 (0.57) TSHRMAPTHCAR2ATMALDH1A1
SCHEMBL8463070 0.91 HCAR2 (0.54) TSHRMAPTHCAR2ATMKEAP1
SCHEMBL7779215 0.91 HCAR2 (0.57) TSHRMAPTHCAR2ATMALDH1A1
SCHEMBL8639055 0.91 HCAR2 (0.57) TSHRMAPTHCAR2ATMALDH1A1
SCHEMBL9618418 0.91 HCAR2 (0.54) TSHRMAPTHCAR2ATMKEAP1
SCHEMBL2808163 0.91 HCAR2 (0.57) TSHRMAPTHCAR2ATMALDH1A1
SCHEMBL18411667 0.91 TSHR (0.45) TSHRMAPTHCAR2ATMKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114381092-A High-temperature thickening vinyl resin and preparation method thereof 江苏博泓新材料科技有限公司 2022-04-22 CN claimed
WO-2019143560-A9 METHODS FOR PROMOTING MITOCHONDRIAL BIOGENESIS IN NEURAL CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-09-12 WO claimed
WO-2019143560-A1 METHODS FOR PROMOTING MITOCHONDRIAL BIOGENESIS IN NEURAL CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-07-25 WO claimed
US-20190111016-A1 METHODS OF TREATING MUSCLE AND LIVER DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-04-18 US claimed
WO-2017147505-A1 METHODS OF TREATING MUSCLE AND LIVER DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-08-31 WO claimed
US-20100240824-A1 POWDER COATING SUSPENSIONS (POWDER SLURRIES) AND POWDER COATING MATERIALS, THEIR PREPARATION AND USE BASF COATINGS AG (DE) 2010-09-23 US claimed
EP-1210379-B1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS UNIV WM MARSH RICE (US) 2007-03-21 EP claimed
EP-1171006-B1 FUNCTIONALIZED POLY(PROPYLENE FUMARATE) AND POLY(PROPYLENE FUMARATE-CO-ETHYLENE GLYCOL) UNIV WM MARSH RICE (US) 2006-03-29 EP claimed
US-6759485-B2 CROSSLINKED ACRYLATED UNSATURATED POLYESTER YIELDS DEGRADATION PRODUCTS NON-TOXIC, METABOLIZED AND EXCRETED BY THE HUMAN KIDNEY; MECHANICAL PROPERTIES, I.E. COMPRESSIVE STRENGTH AND MODULUS; LOW WATER ABSORPTION; GRAFTING IMPLANTS WILLIAM MARSH RICE UNIVERSITY 2004-07-06 US claimed
JP-2002542349-A 2002-12-10 JP claimed
JP-2002542339-A 2002-12-10 JP claimed
EP-1210379-A4 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS UNIV WM MARSH RICE (US) 2002-09-25 EP claimed
EP-1171006-A4 FUNCTIONALIZED POLY(PROPYLENE FUMARATE) AND POLY(PROPYLENE FUMARATE-CO-ETHYLENE GLYCOL) UNIV WM MARSH RICE (US) 2002-09-25 EP claimed
EP-1210379-A1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS Wm. MARSH RICE UNIVERSITY (US) 2002-06-05 EP claimed
EP-1171006-A1 FUNCTIONALIZED POLY(PROPYLENE FUMARATE) AND POLY(PROPYLENE FUMARATE-CO-ETHYLENE GLYCOL) Wm. MARSH RICE UNIVERSITY (US) 2002-01-16 EP claimed
US-6306821-B1 Functionalized poly(propylene fumarate) and poly(propylene fumarate-co-ethylene glycol) WM. MARSH RICE UNIVERSITY 2001-10-23 US claimed
WO-2000063263-A1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS WM. MARSH RICE UNIVERSITY (US) 2000-10-26 WO claimed
WO-2000062630-A1 FUNCTIONALIZED POLY(PROPYLENE FUMARATE) AND POLY(PROPYLENE FUMARATE-CO-ETHYLENE GLYCOL) WM. MARSH RICE UNIVERSITY (US) 2000-10-26 WO claimed
US-4707513-A CROSSLINKED ELASTOMER CORE MONSANTO COMPANY (US) 1987-11-17 US claimed
CN-114381092-A High-temperature thickening vinyl resin and preparation method thereof 江苏博泓新材料科技有限公司 2022-04-22 CN disclosed
US-20200231904-A1 A SOAP BAR BASF PERSONAL CARE AND NUTRITION GMBH (DE) 2020-07-23 US disclosed
EP-3662048-A1 A SOAP BAR BASF SE (DE) 2020-06-10 EP disclosed
CN-110945111-A Soap block 巴斯夫欧洲公司 2020-03-31 CN disclosed
WO-2019143560-A9 METHODS FOR PROMOTING MITOCHONDRIAL BIOGENESIS IN NEURAL CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-09-12 WO disclosed
WO-2019143560-A1 METHODS FOR PROMOTING MITOCHONDRIAL BIOGENESIS IN NEURAL CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-07-25 WO disclosed
US-10336918-B2 Adhesive composition ZEON CORPORATION (JP) 2019-07-02 US disclosed
US-20190111016-A1 METHODS OF TREATING MUSCLE AND LIVER DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-04-18 US disclosed
WO-2019025257-A1 A SOAP BAR BASF SE (DE) 2019-02-07 WO disclosed
US-20180333386-A1 AGENTS USEFUL FOR TREATING FRIEDREICH'S ATAXIA AND OTHER NEURODEGENERATIVE DISEASES IXCHEL PHARMA LLC (US) 2018-11-22 US disclosed
EP-2891694-B1 ADHESIVE AGENT COMPOSITION ZEON CORP (JP) 2018-06-06 EP disclosed
WO-2017147505-A1 METHODS OF TREATING MUSCLE AND LIVER DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-08-31 WO disclosed
US-9469941-B2 Paraben derivatives for preserving cellulosic materials EMPIRE TECHNOLOGY DEVELOPMENT LLC (US) 2016-10-18 US disclosed
US-20150225618-A1 ADHESIVE COMPOSITION ZEON CORPORATION (JP) 2015-08-13 US disclosed
EP-2891694-A1 ADHESIVE AGENT COMPOSITION Zeon Corporation (JP) 2015-07-08 EP disclosed
US-20140206250-A1 ADHESIVE COMPOSITION ZEON CORPORATION (JP) 2014-07-24 US disclosed
EP-2752475-A1 ADHESIVE COMPOSITION Zeon Corporation (JP) 2014-07-09 EP disclosed
US-20130004785-A1 PARABEN DERIVATIVES FOR PRESERVING CELLULOSIC MATERIALS CRESTLINE DIRECT FINANCE, L.P. 2013-01-03 US disclosed
WO-2012149478-A2 AGENTS USEFUL FOR TREATING FRIEDREICH'S ATAXIA AND OTHER NEURODEGENERATIVE DISEASES SERKET PHARMA, LLC (US) 2012-11-01 WO disclosed
EP-1282428-B1 BIOCOMPATIBLE MACROMERS UNIV WM MARSH RICE (US) 2012-07-11 EP disclosed
EP-1812481-B1 BLOCK COPOLYMERS OF POLYCAPROLACTONE AND POLY (PROPYLENE FUMARATE) MAYO FOUNDATION (US) 2012-01-11 EP disclosed
US-7816461-B2 Block copolymers of polycarpolactone and poly (propylene funarate) NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2010-10-19 US disclosed
EP-1194463-B1 POLY(PROPYLENE FUMARATE) CROSS LINKED WITH POLY(ETHYLENE GLYCOL)-DIMETHACRYLATE UNIV WM MARSH RICE (US) 2009-11-11 EP disclosed
US-20080004368-A1 Block Copolymers of Polycarpolactone and Poly (Propylene Funarate) NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2008-01-03 US disclosed
EP-1282428-A4 BIOCOMPATIBLE MACROMERS UNIV WM MARSH RICE (US) 2007-09-05 EP disclosed
EP-1210379-B1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS UNIV WM MARSH RICE (US) 2007-03-21 EP disclosed
EP-1210379-B1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS UNIV WM MARSH RICE (US) 2007-03-21 EP disclosed
US-6884778-B2 Biocompatible macromers WILLIAM MARSH RICE UNIVERSITY (US) 2005-04-26 US disclosed
US-6759485-B2 CROSSLINKED ACRYLATED UNSATURATED POLYESTER YIELDS DEGRADATION PRODUCTS NON-TOXIC, METABOLIZED AND EXCRETED BY THE HUMAN KIDNEY; MECHANICAL PROPERTIES, I.E. COMPRESSIVE STRENGTH AND MODULUS; LOW WATER ABSORPTION; GRAFTING IMPLANTS WILLIAM MARSH RICE UNIVERSITY 2004-07-06 US disclosed
EP-1282428-A1 BIOCOMPATIBLE MACROMERS Wm. MARSH RICE UNIVERSITY (US) 2003-02-12 EP disclosed
EP-1194463-A4 POLY(PROPYLENE FUMARATE) CROSS LINKED WITH POLY(ETHYLENE GLYCOL) UNIV WM MARSH RICE (US) 2002-09-25 EP disclosed
EP-1210379-A4 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS UNIV WM MARSH RICE (US) 2002-09-25 EP disclosed
US-6423790-B1 TISSUE REPLACEMENTS WILLIAM MARSH RICE UNIVERSITY 2002-07-23 US disclosed
EP-1210379-A1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS Wm. MARSH RICE UNIVERSITY (US) 2002-06-05 EP disclosed
US-6384105-B1 INJECTABLE, IN SITU CROSSLINKABLE, BIODEGRADABLE CARRIER FOR BIOACTIVE DRUG DELIVERY WILLIAM MARSH RICE UNIVERSITY 2002-05-07 US disclosed
EP-1194463-A1 POLY(PROPYLENE FUMARATE) CROSS LINKED WITH POLY(ETHYLENE GLYCOL) Wm. MARSH RICE UNIVERSITY (US) 2002-04-10 EP disclosed
US-20020028189-A1 Biocompatible macromers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-03-07 US disclosed
US-20020022676-A1 Poly(Propylene Fumarate) cross linked with Poly(Ethylene Glycol) NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-02-21 US disclosed
WO-2001085180-A1 BIOCOMPATIBLE MACROMERS WM. MARSH RICE UNIVERSITY (US) 2001-11-15 WO disclosed
WO-2000063268-A1 POLY(PROPYLENE FUMARATE) CROSS LINKED WITH POLY(ETHYLENE GLYCOL) WM. MARSH RICE UNIVERSITY (US) 2000-10-26 WO disclosed
WO-2000063263-A1 BIODEGRADABLE POLY(PROPYLENE FUMARATE) NETWORKS CROSS LINKED WITH POLY(PROPYLENE FUMARATE)-DIACRYLATE MACROMERS WM. MARSH RICE UNIVERSITY (US) 2000-10-26 WO disclosed
EP-0786495-B1 Thermoplastic polyester resin stretched film OJI YUKA SYNT PAPER CO LTD (JP) 2000-04-12 EP disclosed
US-5677055-A POLYESTER RESIN, MODIFIED OLEFIN OBTAINED BY GRAFT POLYMERIZING ALPHA, BETA-UNSATURATED CARBOXYLATE MONOMER CONTAINING HYDROXYL GROUPS AND AROMATIC VINYL MONOMER ONTO OLEFIN, POLYETHYLENE, EPOXY RESIN; RECORDING PAPER SUPPORT OJI-YUKA SYNTHETIC PAPER CO., LTD. (JP) 1997-10-14 US disclosed
EP-0786495-A2 Thermoplastic polyester resin stretched film OJI-YUKA SYNTHETIC PAPER CO., LTD. (JP) 1997-07-30 EP disclosed
EP-0612773-B1 Thermoplastic resin composition and process for preparing modified polyolefin type resin MITSUBISHI CHEM CORP (JP) 1996-12-27 EP disclosed
US-5424359-A Aromatic vinyl polymer having alpha, beta-unsaturated carboxylate having a hydroxyl group grafted onto it, and saturated polyester MITSUBISHI PETROCHEMICAL CO., LTD. (JP) 1995-06-13 US disclosed
US-5420187-A Dispersant and monomer with polymerization catalyst and pigment TOYO INK MANUFACTURING CO., LTD. (JP) 1995-05-30 US disclosed
EP-0612773-A1 Thermoplastic resin composition and process for preparing modified polyolefin type resin MITSUBISHI CHEMICAL CORPORATION (JP) 1994-08-31 EP disclosed
EP-0051471-B2 TOUGH THERMOPLASTIC NYLON COMPOSITIONS AND PROCESSES FOR PREPARING THEM MONSANTO COMPANY (US) 1991-11-21 EP disclosed
US-4707513-A CROSSLINKED ELASTOMER CORE MONSANTO COMPANY (US) 1987-11-17 US disclosed
US-4584344-A POLYAMIDE MATRIX AND SHELL-CORE POLYMER CONTAINING CROSSLINKED ELAATOMER CORE AND SHELL OF UNSATURATED ACID, AND STYRENE MONSANTO COMPANY (US) 1986-04-22 US disclosed
EP-0051471-B1 TOUGH THERMOPLASTIC NYLON COMPOSITIONS AND PROCESSES FOR PREPARING THEM MONSANTO COMPANY (US) 1985-06-05 EP disclosed
US-4017448-A Transparent pigment dispersion process CELANESE COATINGS & SPECIALTIES COMPANY (US) 1977-04-12 US disclosed
US-4009684-A Water soluble polymers useful in the preparation of novel animal litter NATIONAL PATENT DEVELOPMENT CORPORATION (US) 1977-03-01 US disclosed
US-3990381-A Hydrophilic polymer coating for underwater structures NATIONAL PATENT DEVELOPMENT CORPORATION (US) 1976-11-09 US disclosed
US-3990381-A Hydrophilic polymer coating for underwater structures NATIONAL PATENT DEVELOPMENT CORPORATION (US) 1976-11-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180333386-A1 AGENTS USEFUL FOR TREATING FRIEDREICH'S ATAXIA AND OTHER NEURODEGENERATIVE DISEASES CLN6, NLN, HTT TSHR 4179/4885MAPT 87/4885HCAR2 3305/4885
US-20080004368-A1 Block Copolymers of Polycarpolactone and Poly (Propylene Funarate) PLOD1, FGB, PLOD2 TSHR 4476/4885MAPT 3085/4885HCAR2 776/4885
US-20190111016-A1 METHODS OF TREATING MUSCLE AND LIVER DISORDERS CKMT1A; CKMT1B, CPT1B, GLS2 TSHR 2836/4885MAPT 2856/4885HCAR2 2186/4885
US-20130004785-A1 PARABEN DERIVATIVES FOR PRESERVING CELLULOSIC MATERIALS CDC73, MGAM, PAXBP1 TSHR 4831/4885MAPT 3627/4885HCAR2 4701/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.