SCHEMBL28082074

SCHEMBL28082074

O=C(O)Cc1ccnc(N2CCCC2)n1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.49
CDC7 O00311 1/20 0.49
ACHE P22303 8/20 0.49
ALDH1A1 P00352 3/20 0.43
GBA1 P04062 1/20 0.41
PKM P14618 1/20 0.41
PANK3 Q9H999 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTPN11 Q06124 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
AOC3 Q16853 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20425054 0.84 ACHE (0.60) ACHEGBA1PANK3KDM4EPTPN11
SCHEMBL28059125 0.79 ACHE (0.46) MAPK8CDC7ACHEGBA1POLB
SCHEMBL21715629 0.77 ACHE (0.47) MAPK8CDC7ACHEGBA1
SCHEMBL15599258 0.76 ACHE (0.46) MAPK8CDC7ACHEGBA1POLB
SCHEMBL28070878 0.76 MAPK8 (0.52) MAPK8CDC7ACHEALDH1A1GBA1
SCHEMBL6502025 0.75 CTSB (0.45) ALDH1A1KDM4ETDP1POLB
SCHEMBL28087268 0.74 MAPK8 (0.54) MAPK8CDC7ACHEALDH1A1GBA1
SCHEMBL27905441 0.74 L3MBTL1 (0.35) ALDH1A1KDM4ETDP1POLB
SCHEMBL1992408 0.74 ACHE (0.48) ACHEPANK3KDM4EAOC3
SCHEMBL31421576 0.73 ACHE (0.43) ACHEAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814049-B Fused tricyclic imdazole derivatives as TNF active regulator UCB生物制药私人有限公司 2019-03-12 CN disclosed
CN-105814049-A Fused tricyclic imidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed