SCHEMBL28085545

SCHEMBL28085545

COc1ccc(-c2c(Nc3ccc(NC(C)=O)cc3)c3ccccc3oc2=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.58
KDM4E B2RXH2 3/20 0.53
ESR1 P03372 3/20 0.50
MAPT P10636 5/20 0.49
TSHR P16473 5/20 0.49
ALDH1A1 P00352 4/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
MAPK1 P28482 1/20 0.49
HPGD P15428 2/20 0.48
RAB9A P51151 2/20 0.48
HSD17B10 Q99714 2/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
GAA P10253 1/20 0.47
NPC1 O15118 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28832577 0.86 ESR1 (0.65) MAOBKDM4EESR1MAPTALDH1A1
SCHEMBL28085659 0.84 ESR1 (0.58) MAOBKDM4EESR1MAPTALDH1A1
SCHEMBL28085701 0.80 MAOB (0.56) MAOBKDM4EESR1MAPTALDH1A1
SCHEMBL28085657 0.76 MAOB (0.52) MAOBKDM4EESR1MAPTALDH1A1
SCHEMBL28085670 0.74 ESR1 (0.73) ESR1MAPTMEN1KMT2ANPC1
SCHEMBL11485562 0.74 MAOB (1.00) MAOBKDM4EMAPTALDH1A1MEN1
Flavonol SCHEMBL7691888 0.73 KDM4E (0.72) MAOBKDM4EMAPTTSHRALDH1A1
SCHEMBL10001286 0.73 SMN1; SMN2 (0.67) KDM4EMAPTTSHRALDH1A1MEN1
SCHEMBL28085548 0.73 ESR1 (0.73) KDM4EESR1MAPTALDH1A1MEN1
SCHEMBL7117054 0.72 MAOB (0.72) MAOBKDM4EMAPTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed