SCHEMBL28085548

SCHEMBL28085548

CCOc1ccc(Nc2c(-c3ccc(OC)cc3)c(=O)oc3cc(O)ccc23)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.73
NPC1 O15118 2/20 0.61
MAPT P10636 3/20 0.49
MEN1 O00255 1/20 0.49
TNKS O95271 1/20 0.49
TP53 P04637 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.49
TNKS2 Q9H2K2 1/20 0.49
NOD2 Q9HC29 1/20 0.49
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085670 0.88 ESR1 (0.73) ESR1NPC1MAPTMEN1TNKS
SCHEMBL28085534 0.87 ESR1 (0.57) ESR1
SCHEMBL28085659 0.86 ESR1 (0.58) ESR1MAPTCYP3A4CYP2C19ALDH1A1
SCHEMBL28085726 0.84 NPC1 (0.64) ESR1NPC1MAPTMEN1TNKS
SCHEMBL5557246 0.78 NPC1 (0.72) ESR1NPC1MAPTMEN1TNKS
SCHEMBL5427914 0.77 NPC1 (1.00) ESR1NPC1MAPTMEN1TNKS
SCHEMBL28085538 0.76 ESR1 (0.54) ESR1NPC1MAPTMEN1KMT2A
SCHEMBL6690691 0.74 ALDH1A1 (0.75) NPC1MAPTMEN1CYP2C9CYP2C19
SCHEMBL5084963 0.74 NPC1 (0.73) ESR1NPC1MAPTMEN1TNKS
SCHEMBL28832577 0.73 ESR1 (0.65) ESR1MAPTMEN1TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed