SCHEMBL28085538

SCHEMBL28085538

COc1ccc(-c2c(Nc3ccc(C)c(O)c3)c3ccc(OCc4ccccc4)cc3oc2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.54
MAOB P27338 5/20 0.51
ACHE P22303 3/20 0.51
CYP19A1 P11511 2/20 0.49
NPC1 O15118 4/20 0.49
MAOA P21397 2/20 0.48
RAB9A P51151 3/20 0.48
CASP3 P42574 2/20 0.48
SENP8 Q96LD8 2/20 0.48
SENP7 Q9BQF6 2/20 0.48
SENP6 Q9GZR1 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085726 0.87 NPC1 (0.64) ESR1MAOBNPC1RAB9AMAPT
SCHEMBL28085534 0.86 ESR1 (0.57) ESR1MAOBACHECYP19A1MAOA
SCHEMBL28085547 0.83 KDM4E (0.58) ESR1MAOBACHECYP19A1MAOA
SCHEMBL28085675 0.81 MAOB (0.65) MAOBACHECYP19A1NPC1MAOA
SCHEMBL28085548 0.76 ESR1 (0.73) ESR1NPC1RAB9AKDM4EALDH1A1
SCHEMBL28085670 0.74 ESR1 (0.73) ESR1NPC1MAPTMEN1KMT2A
SCHEMBL28085539 0.73 CYP19A1 (0.59) ESR1MAOBACHECYP19A1NPC1
SCHEMBL6823769 0.71 MAOB (0.53) ESR1MAOBACHECYP19A1NPC1
SCHEMBL28085659 0.71 ESR1 (0.58) ESR1MAOBRAB9ATDP1KDM4E
SCHEMBL5084963 0.70 NPC1 (0.73) ESR1MAOBCYP19A1NPC1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed