SCHEMBL28085534

SCHEMBL28085534

CCOc1ccc(Nc2c(-c3ccc(OC)cc3)c(=O)oc3cc(OCc4ccccc4)ccc23)cc1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.57
CYP19A1 P11511 3/20 0.52
MAOB P27338 5/20 0.52
ACHE P22303 2/20 0.52
MAOA P21397 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085548 0.87 ESR1 (0.73) ESR1
SCHEMBL28085547 0.86 KDM4E (0.58) ESR1CYP19A1MAOBACHEMAOA
SCHEMBL28085538 0.86 ESR1 (0.54) ESR1CYP19A1MAOBACHEMAOA
SCHEMBL28085659 0.85 ESR1 (0.58) ESR1MAOB
SCHEMBL28085675 0.80 MAOB (0.65) CYP19A1MAOBACHEMAOA
SCHEMBL7115073 0.79 ALDH1A1 (0.56) CYP19A1MAOBACHE
SCHEMBL28085539 0.77 CYP19A1 (0.59) ESR1CYP19A1MAOBACHEMAOA
SCHEMBL28085670 0.75 ESR1 (0.73) ESR1
SCHEMBL6690691 0.75 ALDH1A1 (0.75) MAOBACHE
SCHEMBL28832577 0.73 ESR1 (0.65) ESR1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed