Butaperazine

Butaperazine

SCHEMBL28086241

CCCC(=O)c1ccc2c(c1)N(CCCN1CCN(C)CC1)c1ccccc1S2.CN1CCN(CCCN2c3ccccc3Sc3ccccc32)CC1

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 7/20 0.67
HTR1A P08908 6/20 0.67
DRD2 P14416 6/20 0.67
ADRA2C P18825 6/20 0.67
SLC6A2 P23975 6/20 0.67
HTR2A P28223 6/20 0.67
SLC6A4 P31645 6/20 0.67
ADRA1A P35348 6/20 0.67
DRD3 P35462 6/20 0.67
SLC6A3 Q01959 6/20 0.67
KCNH2 Q12809 6/20 0.67
ADRA2A P08913 5/20 0.67
DRD1 P21728 5/20 0.67
ADRA2B P18089 5/20 0.67
HTR2B P41595 4/20 0.67
HRH3 Q9Y5N1 4/20 0.67
MLNR O43193 2/20 0.67
ESR1 P03372 2/20 0.67
PTGS2 P35354 1/20 0.67
KDM1A O60341 3/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butaperazine SCHEMBL119995 1.00 HRH1 (0.67) HRH1HTR1ADRD2ADRA2CSLC6A2
Butaperazine SCHEMBL29710903 1.00 HRH1 (0.67) HRH1HTR1ADRD2ADRA2CSLC6A2
Butaperazine SCHEMBL31153317 1.00 HRH1 (0.67) HRH1HTR1ADRD2ADRA2CSLC6A2
Butaperazine SCHEMBL120744 0.94 LMNA (0.72) HRH1HTR1ADRD2ADRA2CSLC6A2
Butaperazine SCHEMBL120743 0.94 LMNA (0.72) HRH1HTR1ADRD2ADRA2CSLC6A2
Thioproperazine SCHEMBL13723252 0.90 DRD3 (0.79) HRH1HTR1ADRD2ADRA2CSLC6A2
SCHEMBL18309819 0.88 HRH1 (0.69) HRH1HTR1ADRD2ADRA2CSLC6A2
SCHEMBL141601 0.87 HTR1A (0.86) HRH1HTR1ADRD2ADRA2CSLC6A2
SCHEMBL26837052 0.85 HRH1 (0.69) HRH1HTR1ADRD2ADRA2CSLC6A2
Carphenazine SCHEMBL1458434 0.84 HRH1 (0.81) HRH1HTR1ADRD2ADRA2CSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed