SCHEMBL28089646

SCHEMBL28089646

COCCOc1cc(I)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 5/20 0.50
ALDH1A1 P00352 4/20 0.50
MAPT P10636 3/20 0.50
POLB P06746 2/20 0.50
HPGD P15428 2/20 0.50
MEN1 O00255 1/20 0.50
USP2 O75604 1/20 0.50
CYP2C9 P11712 1/20 0.50
ALOX12 P18054 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
LMNA P02545 2/20 0.38
S1PR4 O95977 2/20 0.38
TRPV1 Q8NER1 1/20 0.37
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15087903 0.91 L3MBTL1 (0.45) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL3105572 0.84 CSNK2A1 (0.47) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL15197103 0.80 TSHR (0.40) L3MBTL1ALDH1A1POLBHPGDCYP2C9
SCHEMBL13861973 0.80 L3MBTL1 (0.75) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL3324595 0.79 ALDH1A1 (0.50) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL2227815 0.79 MAPT (0.50) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL22596995 0.79 L3MBTL1 (0.50) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL22964315 0.79 L3MBTL1 (0.50) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL8265598 0.79 HPGD (0.50) L3MBTL1ALDH1A1MAPTPOLBHPGD
SCHEMBL27819584 0.79 L3MBTL1 (0.50) L3MBTL1ALDH1A1MAPTPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777756-B Heteroaryl compound and its application in drug 广东东阳光药业有限公司 2019-03-01 CN disclosed
CN-105777756-A Heteroaryl compound and application thereof in medicines 广东东阳光药业有限公司 2016-07-20 CN disclosed