SCHEMBL28090659

SCHEMBL28090659

Cc1[nH]ccc1NC(CO)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
CCNT1 O60563 7/20 0.41
CDK9 P50750 7/20 0.41
CDK2 P24941 3/20 0.41
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RIPK1 Q13546 1/20 0.39
JAK3 P52333 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
DYRK3 O43781 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CLK1 P49759 1/20 0.38
CLK3 P49761 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
DYRK2 Q92630 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28090879 1.00 IDO1 (0.43) IDO1TDO2CCNT1CDK9CDK2
SCHEMBL28090877 0.82 MAN2A1 (0.40) EGFRMAN2A1MAN1B1
SCHEMBL431572 0.77 HPGD (0.49) IDO1TDO2CDK2LMNAHPGD
SCHEMBL431571 0.70 NPBWR1 (0.54) CCNT1CDK9LMNAHPGDSMN1; SMN2
SCHEMBL21410829 0.70 JAK3 (0.44) IDO1TDO2LMNARIPK1JAK3
SCHEMBL20095129 0.70 MAPKAPK2 (0.54) IDO1TDO2CDK2LMNARIPK1
SCHEMBL27783713 0.70 MAPKAPK2 (0.54) IDO1TDO2CDK2LMNARIPK1
SCHEMBL430689 0.70 MAPKAPK2 (0.54) IDO1TDO2CDK2LMNARIPK1
SCHEMBL1964723 0.68 ALDH1A1 (0.55) CDK2RIPK1CYP2C9CYP2C19GSK3B
SCHEMBL4110424 0.68 ALDH1A1 (0.55) CDK2RIPK1CYP2C9CYP2C19GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103848833-B Pyrrolo-triazine analog derivative, its preparation method and in application pharmaceutically 上海希迈医药科技有限公司 2016-08-31 CN disclosed