SCHEMBL28094044

SCHEMBL28094044

CC(C)(C)SN=Cc1cc(C(F)(F)F)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.39
IDO1 P14902 2/20 0.36
PDE2A O00408 4/20 0.34
GAA P10253 1/20 0.32
KIF11 P52732 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MPL P40238 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.30
APP P05067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28094043 1.00 BACE1 (0.39) BACE1IDO1PDE2AGAAKIF11
SCHEMBL28093529 0.88 PDE2A (0.37) BACE1IDO1PDE2AGAAKIF11
SCHEMBL28093533 0.88 PDE2A (0.37) BACE1IDO1PDE2AGAAKIF11
SCHEMBL23070808 0.82 NFE2L2 (0.41) GAAMAPT
SCHEMBL23070810 0.82 NFE2L2 (0.41) GAAMAPT
SCHEMBL30608104 0.81 AMY1A (0.34) KDM4EMAPTALDH1A1
SCHEMBL19634050 0.81 KDM4E (0.41) GAAKDM4EMAPTMEN1KMT2A
SCHEMBL28333129 0.78 PDE2A (0.37) PDE2AGAAKIF11SMN1; SMN2
SCHEMBL28333131 0.78 PDE2A (0.37) PDE2AGAAKIF11SMN1; SMN2
SCHEMBL28338194 0.77 AMY1A (0.46) GAAKDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106478497-A Aryl amine derivatives as TTX S blocker 拉夸里亚创药株式会社 2017-03-08 CN disclosed
CN-103249721-B Arylamine Derivatives as TTX-S Blockers 拉夸里亚创药株式会社 2016-10-12 CN disclosed