SCHEMBL28096006

SCHEMBL28096006

CP(=O)(O)Oc1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
KMT2A Q03164 2/20 0.44
CYP2C19 P33261 1/20 0.43
FDPS P14324 3/20 0.42
CHRNB2 P17787 3/20 0.42
CHRNA4 P43681 3/20 0.42
HTT P42858 1/20 0.41
POLB P06746 1/20 0.41
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28219782 0.85 SRC (0.57) SMN1; SMN2LMNATDP1KMT2AFDPS
SCHEMBL27714398 0.82 KMT2A (0.45) SMN1; SMN2LMNATDP1KMT2AFDPS
SCHEMBL4744280 0.81 SMN1; SMN2 (0.45) SMN1; SMN2LMNATDP1KMT2AFDPS
SCHEMBL18301043 0.81 SMN1; SMN2 (0.42) SMN1; SMN2LMNATDP1KMT2AFDPS
SCHEMBL27647649 0.77 FDPS (0.45) SMN1; SMN2LMNATDP1FDPSCHRNB2
SCHEMBL4679260 0.77 FDPS (0.44) SMN1; SMN2LMNATDP1KMT2AFDPS
SCHEMBL4744278 0.77 SMN1; SMN2 (0.47) SMN1; SMN2LMNATDP1KMT2ACHRNB2
SCHEMBL10932461 0.77 SMN1; SMN2 (0.47) SMN1; SMN2LMNATDP1KMT2ACHRNB2
SCHEMBL27998020 0.76 LMNA (0.43) SMN1; SMN2LMNATDP1KMT2ACHRNB2
SCHEMBL27707122 0.76 CYP2C19 (0.53) SMN1; SMN2LMNAKMT2ACYP2C19FDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596985-B 17-hydroxy-17-pentafluoroethyl-estra-4, 9(10) -dien-11-aryl derivatives, method for the production thereof and use thereof for treating diseases 拜耳知识产权有限责任公司 2017-05-24 CN disclosed
CN-106046100-A 17-hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-aryl derivatives, methods for the production thereof and the use thereof for treating diseases 拜耳知识产权有限责任公司 2016-10-26 CN disclosed