SCHEMBL28096097

SCHEMBL28096097

COc1ccc2c(c1)C(=O)C(=Cc1cc(OC)c(OC)c(OC)c1Br)CC2

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.66
BCHE P06276 1/20 0.64
ACHE P22303 1/20 0.64
ALDH1A1 P00352 3/20 0.58
MAPT P10636 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
MAPK1 P28482 1/20 0.58
MAOB P27338 2/20 0.58
CYP19A1 P11511 2/20 0.56
PLA2G1B P04054 1/20 0.56
RAB9A P51151 1/20 0.56
ATG4B Q9Y4P1 1/20 0.56
MAOA P21397 2/20 0.55
CYP26A1 O43174 1/20 0.55
CYP27A1 Q02318 1/20 0.55
MEN1 O00255 1/20 0.52
GAA P10253 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28096102 0.92 BCHE (0.74) EGFRBCHEACHEALDH1A1MAPT
SCHEMBL28096393 0.83 BCHE (0.61) EGFRBCHEACHEALDH1A1MAPT
SCHEMBL28095988 0.82 BCHE (0.64) EGFRBCHEACHEALDH1A1MAPT
SCHEMBL28096418 0.76 MAOA (0.68) ALDH1A1MAPTSMN1; SMN2MAOBCYP19A1
SCHEMBL28096395 0.76 MAPT (0.80) BCHEACHEALDH1A1MAPTSMN1; SMN2
SCHEMBL3502646 0.76 MAOB (0.85) ACHEALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL13254636 0.76 MAOB (0.85) ACHEALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL28833618 0.74 BCHE (0.74) BCHEACHEALDH1A1MAPTSMN1; SMN2
SCHEMBL5692075 0.74 ALDH1A1 (0.75) ALDH1A1MAPTSMN1; SMN2MAPK1MAOB
SCHEMBL5691865 0.74 NFE2L2 (0.67) ALDH1A1MAPTSMN1; SMN2MAPK1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106278857-A α, β unsaturated carbonyl tetralone derivative and application thereof 武汉理工大学 2017-01-04 CN claimed
CN-106008324-A Alpha,beta-unsaturated compounds and application thereof 武汉理工大学 2016-10-12 CN claimed
CN-106278857-A α, β unsaturated carbonyl tetralone derivative and application thereof 武汉理工大学 2017-01-04 CN disclosed
CN-106008324-A Alpha,beta-unsaturated compounds and application thereof 武汉理工大学 2016-10-12 CN disclosed