SCHEMBL28096102

SCHEMBL28096102

COc1ccc2c(c1)CCC(=Cc1cc(OC)c(OC)c(OC)c1Br)C2=O

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.74
ACHE P22303 1/20 0.74
EGFR P00533 2/20 0.74
ALDH1A1 P00352 3/20 0.69
MAPT P10636 3/20 0.69
SMN1; SMN2 Q16637 3/20 0.69
MAPK1 P28482 1/20 0.69
CYP26A1 O43174 2/20 0.65
CYP27A1 Q02318 2/20 0.65
ABCB1 P08183 1/20 0.59
CYP24A1 Q07973 3/20 0.57
MIF P14174 2/20 0.57
RAB9A P51151 2/20 0.57
PLA2G1B P04054 1/20 0.57
ATG4B Q9Y4P1 1/20 0.57
KDM4E B2RXH2 1/20 0.56
NPC1 O15118 1/20 0.56
HPGD P15428 1/20 0.56
NFKB1 P19838 1/20 0.56
NFKB2 Q00653 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28096097 0.92 EGFR (0.66) BCHEACHEEGFRALDH1A1MAPT
SCHEMBL28833618 0.82 BCHE (0.74) BCHEACHEALDH1A1MAPTSMN1; SMN2
SCHEMBL9619624 0.82 ALDH1A1 (0.79) ALDH1A1MAPTSMN1; SMN2MAPK1CYP26A1
SCHEMBL9619490 0.82 NFE2L2 (0.71) ALDH1A1MAPTSMN1; SMN2MAPK1CYP26A1
SCHEMBL28096393 0.81 BCHE (0.61) BCHEACHEEGFRALDH1A1MAPT
SCHEMBL28096395 0.77 MAPT (0.80) BCHEACHEALDH1A1MAPTSMN1; SMN2
SCHEMBL28096059 0.76 CYP26A1 (0.67) ALDH1A1MAPTSMN1; SMN2MAPK1CYP26A1
SCHEMBL17313263 0.75 CYP26A1 (0.71) ALDH1A1MAPTSMN1; SMN2MAPK1CYP26A1
SCHEMBL17313264 0.75 CYP26A1 (0.71) ALDH1A1MAPTSMN1; SMN2MAPK1CYP26A1
SCHEMBL6958968 0.75 MIF (0.85) BCHEACHEALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106278857-A α, β unsaturated carbonyl tetralone derivative and application thereof 武汉理工大学 2017-01-04 CN claimed
CN-106008324-A Alpha,beta-unsaturated compounds and application thereof 武汉理工大学 2016-10-12 CN claimed
CN-106278857-A α, β unsaturated carbonyl tetralone derivative and application thereof 武汉理工大学 2017-01-04 CN disclosed
CN-106008324-A Alpha,beta-unsaturated compounds and application thereof 武汉理工大学 2016-10-12 CN disclosed