SCHEMBL28096890

SCHEMBL28096890

COc1cc(Br)ccc1OC(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
TSHR P16473 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP3A4 P08684 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA7 P43166 1/20 0.46
TPMT P51580 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
SLC9A1 P19634 1/20 0.45
ALDH1A1 P00352 4/20 0.44
HPGD P15428 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1603755 0.84 TSHR (0.62) MAPTTSHRSMN1; SMN2ALDH1A1KDM4E
Methyl Alcohol SCHEMBL28799088 0.82 CA2 (0.52) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL29419589 0.82 CA2 (0.56) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL20509 0.82 CA2 (0.56) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL2829108 0.82 ALDH1A1 (0.44) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL7364004 0.81 ALDH1A1 (0.46) MAPTTSHRCYP1A2CYP2C9CYP2C19
Acetic Acid SCHEMBL27710642 0.81 CA12 (0.49) MAPTTSHRCYP1A2CYP2C9CYP2C19
Formaldehyde SCHEMBL23581083 0.81 CA2 (0.50) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL1256865 0.80 CA2 (0.54) MAPTTSHRCYP1A2CYP2C9CYP2C19
SCHEMBL3325627 0.80 TNFSF11 (0.55) MAPTTSHRCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110036014-B Compound with AXL inhibitory activity and preparation and application thereof 中国科学院上海药物研究所 2021-09-07 CN disclosed
CN-105884695-A Heterocyclic derivate tyrosine kinase inhibitor 山东轩竹医药科技有限公司 2016-08-24 CN disclosed