SCHEMBL28097258

SCHEMBL28097258

NC(=O)Oc1ccc(F)cc1CBr

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.41
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 1/20 0.35
SLC9A1 P19634 2/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
PTPN1 P18031 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
NTRK1 P04629 1/20 0.34
MPO P05164 1/20 0.33
PARP1 P09874 1/20 0.33
HDAC3 O15379 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27469437 0.87 PKM (0.39) PKMFFAR1FFAR4MEN1KMT2A
SCHEMBL28055980 0.87 PKM (0.37) PKMFFAR1FFAR4MEN1KMT2A
SCHEMBL28615069 0.85 PKM (0.38) PKMFFAR1FFAR4MEN1KMT2A
SCHEMBL27936436 0.85 FFAR1 (0.40) PKMFFAR1FFAR4CYP3A4CYP2C19
SCHEMBL28963024 0.80 PKM (0.39) PKMFFAR1FFAR4MEN1KMT2A
SCHEMBL11712958 0.79 MEN1 (0.39) MEN1KMT2AALDH1A1
SCHEMBL27850278 0.78 CYP3A4 (0.43) FFAR1FFAR4KMT2ACYP3A4CYP2C19
SCHEMBL27585418 0.78 MPO (0.37) PKMFFAR1FFAR4MEN1KMT2A
SCHEMBL16685788 0.77 PKM (0.56) PKMFFAR1FFAR4MEN1KMT2A
SCHEMBL6172318 0.77 CES2 (0.45) MEN1KMT2ACYP3A4CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110498759-A The synthetic method of isoindoline ketone compound TIANJIN RUILING CHEMICAL CO LTD 2019-11-26 CN disclosed
CN-107250126-B Long-acting dipeptidyl peptidase-IV inhibitor, application and preparation method thereof 四川科伦博泰生物医药股份有限公司 2019-10-25 CN disclosed
CN-109415355-A Benzdioxan derivative and its medicinal usage 奥赖恩公司 2019-03-01 CN disclosed
CN-109265443-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-01-25 CN disclosed
CN-107250126-A Long-acting dipeptidyl peptidase-IV inhibitor, application and preparation method thereof 四川科伦博泰生物医药股份有限公司 2017-10-13 CN disclosed
CN-104230827-B 1-(aryl methyl) quinazoline-2,4 (1H, 3H)-diketone is as PARP inhibitor and application thereof 南京英派药业有限公司 2016-10-26 CN disclosed