SCHEMBL28055980

SCHEMBL28055980

NC(=O)Oc1cc(F)ccc1CBr

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.37
IDO1 P14902 2/20 0.36
AGXT P21549 2/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MPO P05164 2/20 0.35
SLC6A4 P31645 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
AKR1A1 P14550 1/20 0.35
AKR1B1 P15121 1/20 0.35
PTPN1 P18031 1/20 0.34
ALDH1A1 P00352 1/20 0.34
FFAR1 O14842 2/20 0.34
FFAR4 Q5NUL3 2/20 0.34
MAPK14 Q16539 2/20 0.34
MAOB P27338 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27585418 0.87 MPO (0.37) PKMIDO1AGXTHDAC3HDAC1
SCHEMBL28097258 0.87 PKM (0.41) PKMHDAC3HDAC1HDAC2HDAC6
SCHEMBL27726752 0.85 IDO1 (0.37) PKMIDO1AGXTHDAC3HDAC1
Hydrochloric Acid SCHEMBL27862891 0.83 IDO1 (0.39) PKMIDO1AGXTHDAC3HDAC1
SCHEMBL6650657 0.83 CYP4F2 (0.44) PKMHDAC3HDAC1HDAC2HDAC6
SCHEMBL28963048 0.80 MEN1 (0.36) PKMHDAC3HDAC1HDAC2HDAC6
SCHEMBL28963079 0.79 LMNA (0.38) PKMHDAC3HDAC1HDAC2HDAC6
SCHEMBL11712958 0.79 MEN1 (0.39) MEN1KMT2AALDH1A1
SCHEMBL27469437 0.78 PKM (0.39) PKMMPOSLC6A4MEN1KMT2A
SCHEMBL27524200 0.77 FFAR1 (0.46) PKMMEN1KMT2AALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105530932-B Primary formamide as BTK inhibitor 艾伯维公司 2019-09-27 CN disclosed
CN-108697684-A The conditioning agent of chemokine receptors 凯莫森特里克斯股份有限公司 2018-10-23 CN disclosed
CN-104230827-B 1-(aryl methyl) quinazoline-2,4 (1H, 3H)-diketone is as PARP inhibitor and application thereof 南京英派药业有限公司 2016-10-26 CN disclosed
CN-105530932-A Primary carboxamides as BIK inhibitors ABBVIE INC 2016-04-27 CN disclosed