SCHEMBL28097398

SCHEMBL28097398

COc1cc(C=NO)cc(Cc2cc(OC)c(OC)c(Br)c2Br)c1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.54
CA2 P00918 7/20 0.54
CA4 P22748 5/20 0.54
CA6 P23280 5/20 0.54
ALDH1A1 P00352 6/20 0.52
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
HTT P42858 4/20 0.52
HPGD P15428 3/20 0.52
HSD17B10 Q99714 2/20 0.51
MAPK1 P28482 1/20 0.51
CYP1A2 P05177 3/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2C19 P33261 3/20 0.46
LMNA P02545 3/20 0.46
MAPT P10636 3/20 0.46
CYP2D6 P10635 1/20 0.46
PKM P14618 2/20 0.45
HSP90AA1 P07900 1/20 0.45
XBP1 P17861 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27785866 0.79 CA2 (0.79) CA1CA2CA4CA6CYP3A4
SCHEMBL21264324 0.77 HSD17B10 (0.59) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL3471747 0.77 HPGD (0.59) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL3471744 0.77 HPGD (0.59) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL15463039 0.77 HPGD (0.59) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL12120526 0.76 HSD17B10 (0.75) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL28097340 0.74 CA1 (0.62) CA1CA2CA4CA6CYP1A2
SCHEMBL22824610 0.73 ALDH1A1 (0.54) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL10050296 0.71 ALDH1A1 (0.52) ALDH1A1MEN1KMT2AHTTHPGD
SCHEMBL30393930 0.71 ALDH1A1 (0.52) ALDH1A1MEN1KMT2AHTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106278941-A Nine kinds of PTP1B inhibitor and synthesis thereof and application 南通中国科学院海洋研究所海洋科学与技术研究发展中心 2017-01-04 CN claimed
CN-106278941-B Nine kinds of PTP1B inhibitor and its synthesis and application 南通中国科学院海洋研究所海洋科学与技术研究发展中心 2018-04-17 CN disclosed
CN-106278941-A Nine kinds of PTP1B inhibitor and synthesis thereof and application 南通中国科学院海洋研究所海洋科学与技术研究发展中心 2017-01-04 CN disclosed