SCHEMBL2809868

SCHEMBL2809868

C#Cc1cccc(C)c1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
TRPA1 O75762 2/20 0.56
GABRA1 P14867 1/20 0.48
GABRB2 P47870 1/20 0.48
ATM Q13315 2/20 0.44
HPGD P15428 3/20 0.42
HSD17B10 Q99714 3/20 0.42
KDM4E B2RXH2 3/20 0.42
TSHR P16473 2/20 0.38
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 1/20 0.36
CA2 P00918 3/20 0.36
CA1 P00915 2/20 0.36
RECQL P46063 2/20 0.36
LMNA P02545 2/20 0.36
ALOX15 P16050 2/20 0.36
ADAMTS4 O75173 1/20 0.36
EGFR P00533 1/20 0.36
FYN P06241 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1808224 0.78 ALDH1A1 (0.55) ALDH1A1TRPA1HPGDHSD17B10KDM4E
SCHEMBL6273994 0.77 ALDH1A1 (0.56) ALDH1A1TRPA1GABRA1GABRB2ATM
SCHEMBL2642471 0.77 TSHR (0.60) ALDH1A1TRPA1GABRA1GABRB2ATM
SCHEMBL2809871 0.77 TRPA1 (0.50) ALDH1A1TRPA1ATMHPGDHSD17B10
SCHEMBL5974541 0.76 TRPA1 (0.42) ALDH1A1TRPA1GABRA1GABRB2ATM
SCHEMBL2813180 0.76 ALDH1A1 (0.54) ALDH1A1TRPA1GABRA1GABRB2ATM
SCHEMBL29463601 0.75
SCHEMBL233965 0.75
SCHEMBL4948998 0.74 TSHR (0.39) ALDH1A1TRPA1GABRA1GABRB2ATM
SCHEMBL64141 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B ALDH1A1 401/4885TRPA1 819/4885GABRA1 2372/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 ALDH1A1 1480/4885TRPA1 1210/4885GABRA1 4045/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.