SCHEMBL2809871

SCHEMBL2809871

C#Cc1cccc(O)c1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.50
ATM Q13315 1/20 0.50
ALDH1A1 P00352 6/20 0.36
CA2 P00918 4/20 0.36
TDP1 Q9NUW8 3/20 0.36
LMNA P02545 3/20 0.36
HPGD P15428 3/20 0.36
ALOX15 P16050 3/20 0.36
HSD17B10 Q99714 3/20 0.36
CA1 P00915 3/20 0.36
EGFR P00533 2/20 0.36
FYN P06241 2/20 0.36
MMP9 P14780 2/20 0.36
RECQL P46063 2/20 0.36
ADAMTS4 O75173 1/20 0.36
MMP2 P08253 1/20 0.36
MMP8 P22894 1/20 0.36
CA6 P23280 1/20 0.36
CDK2 P24941 1/20 0.36
MMP12 P39900 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13981332 0.79 TRPA1 (0.36) TRPA1ATMALDH1A1TDP1KDM4E
SCHEMBL1808224 0.78 ALDH1A1 (0.55) TRPA1ALDH1A1CA2TDP1LMNA
SCHEMBL29451048 0.77 TRPA1 (0.50) TRPA1ATMALDH1A1CA2TDP1
SCHEMBL16954573 0.77 TRPA1 (0.50) TRPA1ATMALDH1A1CA2TDP1
SCHEMBL2137032 0.77 TRPA1 (0.50) TRPA1ATMALDH1A1CA2TDP1
SCHEMBL1631930 0.77 TRPA1 (0.50) TRPA1ATMALDH1A1CA2TDP1
SCHEMBL2809868 0.77 ALDH1A1 (0.56) TRPA1ATMALDH1A1CA2TDP1
SCHEMBL27309120 0.77 CYP1A1 (0.40) TRPA1ATMALDH1A1TDP1HPGD
SCHEMBL5974541 0.76 TRPA1 (0.42) TRPA1ATMALDH1A1CA2CA1
SCHEMBL2813183 0.76 TRPA1 (0.48) TRPA1ATMALDH1A1CA2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734686-B Catalytic synthesis method of 2-substituted benzofuran compound 浙江万里学院 2022-07-01 CN claimed
CN-109734686-B Catalytic synthesis method of 2-substituted benzofuran compound 浙江万里学院 2022-07-01 CN disclosed
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
CN-101868444-A Acetylenic compound, salt thereof, condensate thereof, and composition thereof FUJIFILM CORP 2010-10-20 CN disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
CN-101808982-A Acetylene compound FUJIFILM CORP 2010-08-18 CN disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-0728742-B1 Novel retinoids HOFFMANN LA ROCHE (CH) 1999-10-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B TRPA1 819/4885ATM 1160/4885ALDH1A1 401/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 TRPA1 1210/4885ATM 1200/4885ALDH1A1 1480/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.