SCHEMBL28099443

SCHEMBL28099443

CCOC(=O)c1cc2ccccc2n1CCC#N

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.65
CRHBP P24387 1/20 0.65
CRHR2 Q13324 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
NOD2 Q9HC29 6/20 0.61
NOD1 Q9Y239 6/20 0.61
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
F10 P00742 2/20 0.55
CNR2 P34972 4/20 0.53
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
ALDH1A1 P00352 4/20 0.48
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111591 0.93 KDM4E (0.63) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL30585515 0.87 NOD2 (0.64) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL1392918 0.87 NOD2 (0.64) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL7880746 0.87 MTNR1A (0.62) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL1979481 0.85 SMN1; SMN2 (0.48) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL7688465 0.85 CNR2 (0.52) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL6752352 0.84 KDM4E (0.71) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL18322286 0.83 KDM4E (0.73) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL13742183 0.83 KDM4E (0.70) KDM4ECRHBPCRHR2SMN1; SMN2NOD2
SCHEMBL30489155 0.83 KDM4E (0.73) KDM4ECRHBPCRHR2SMN1; SMN2NOD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103992326-B Indole hexahydropyrazine quinazolinone anti-tumor compounds and preparation method thereof 中国人民解放军第二军医大学 2016-09-28 CN claimed
CN-103992326-B Indole hexahydropyrazine quinazolinone anti-tumor compounds and preparation method thereof 中国人民解放军第二军医大学 2016-09-28 CN disclosed