SCHEMBL28099665

SCHEMBL28099665

C#Cc1c(C(=O)c2ccccc2)cc(F)c(F)c1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
ADORA1 P30542 1/20 0.40
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40
ATM Q13315 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDE4A P27815 1/20 0.38
HPGD P15428 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PTPN22 Q9Y2R2 2/20 0.38
PTPRC P08575 1/20 0.38
PTPN9 P43378 1/20 0.38
PTPN11 Q06124 1/20 0.38
CNR2 P34972 4/20 0.38
CNR1 P21554 2/20 0.38
AKR1C3 P42330 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28133754 0.82 PDE4A (0.44) NR1H2NR1H3ADORA1HSD17B1HSD17B2
SCHEMBL4150417 0.72 RAB9A (0.52) HSD17B1HSD17B2ATMTDP1L3MBTL1
SCHEMBL1505897 0.72 TTR (0.53) NR1H2NR1H3ADORA1ATMTDP1
SCHEMBL8769335 0.72 AKR1C3 (0.48) HSD17B1HSD17B2ATMTDP1L3MBTL1
SCHEMBL5502719 0.70 BCAT2 (0.41) ALDH1A1PTPN22PTPRCPTPN9PTPN11
SCHEMBL934810 0.69 AKR1C3 (0.59) NR1H2NR1H3ADORA1ATMTDP1
SCHEMBL10647658 0.69 BCL2 (0.53) HSD17B1HSD17B2ATMTDP1L3MBTL1
SCHEMBL15793447 0.68 MAPT (0.50) ADORA1ATMTDP1L3MBTL1ALDH1A1
SCHEMBL10644840 0.68 HPGD (0.48) ATMTDP1L3MBTL1PDE4AHPGD
SCHEMBL7557427 0.68 AKR1C3 (0.48) ATMTDP1L3MBTL1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105940036-A POLYMERIC MATERIALS 威格斯制造有限公司 2016-09-14 CN disclosed